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ADR-851 free base
🥰Excellent
Catalog No. T23642Cas No. 138559-56-5
Alias ADR851 free base, ADR 851 free base
ADR-851 free base (ADR 851 free base) is a 5-HT3 receptor antagonist and a novel antiemetic with analgesic activity.
ADR-851 free base
🥰Excellent
Purity: 98.32%
Catalog No. T23642Alias ADR851 free base, ADR 851 free baseCas No. 138559-56-5
ADR-851 free base (ADR 851 free base) is a 5-HT3 receptor antagonist and a novel antiemetic with analgesic activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 5 mg | $722 | In Stock | |
| 10 mg | $987 | In Stock | |
| 25 mg | $1,520 | In Stock | |
| 50 mg | $1,980 | In Stock |
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CitedSelect Batch
Purity:98.32%
ee:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | ADR-851 free base (ADR 851 free base) is a 5-HT3 receptor antagonist and a novel antiemetic with analgesic activity. |
| In vivo | Male Sprague-Dawley rats were injected intraperitoneally with ADR-851 (0.1-10 mg/kg), and the ADR-851 isoforms were not analgesic in either the thermal or mechanical tests; ADR-851R produced significant analgesia in the formalin test at doses of 3 mg/kg and 10 mg/kg.[1] |
| Alias | ADR851 free base, ADR 851 free base |
| Molecular Weight | 295.77 |
| Formula | C14H18ClN3O2 |
| Cas No. | 138559-56-5 |
| Smiles | C(NC[C@@H]1CCCN1)(=O)C2=C3C(=C(N)C(Cl)=C2)CCO3 |
| Relative Density. | 1.314 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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