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BZAD01

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Catalog No. T25196Cas No. 305339-41-7
Alias BZAD-01, BZAD 01

BZAD01 is a selective NMDA NR1A/2B receptor antagonist.

BZAD01

BZAD01

🥰Excellent
Purity: 99.78%
Catalog No. T25196Alias BZAD-01, BZAD 01Cas No. 305339-41-7
BZAD01 is a selective NMDA NR1A/2B receptor antagonist.
Pack SizePriceAvailabilityQuantity
2 mg$39In Stock
5 mg$77In Stock
10 mg$127In Stock
25 mg$255In Stock
50 mg$397In Stock
100 mg$658In Stock
200 mg$919In Stock
1 mL x 10 mM (in DMSO)$108In Stock
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Purity:99.78%
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Product Introduction

Bioactivity
Description
BZAD01 is a selective NMDA NR1A/2B receptor antagonist.
In vivo
Parkinsonism was induced by microinjection of the toxin, 6-hydroxydopamine (6-OHDA) into the medial forebrain bundle (MFB) of 40 Sprague-Dawley rats. Parkinsonism and the efficacy of drugs were assessed using a battery of behavioural tests including balance beam, apomorphine-induced rotation, body axis bias or "curling", head position bias and disengage sensorimotor latency test. The main effects were that BZAD01 co-administration prevented chronic levodopa-induced potentiation of apomorphine rotation. However levodopa-treated rats were slower than either controls or BZAD-01-treated rats in the locomotor test[2].
AliasBZAD-01, BZAD 01
Chemical Properties
Molecular Weight362.27
FormulaC16H12F6N2O
Cas No.305339-41-7
SmilesFC(F)(F)Oc1ccc(cc1)C(=N)NCc1ccccc1C(F)(F)F
Relative Density.1.34 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 55 mg/ml (151.82 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.7604 mL13.8019 mL27.6037 mL138.0186 mL
5 mM0.5521 mL2.7604 mL5.5207 mL27.6037 mL
10 mM0.2760 mL1.3802 mL2.7604 mL13.8019 mL
20 mM0.1380 mL0.6901 mL1.3802 mL6.9009 mL
50 mM0.0552 mL0.2760 mL0.5521 mL2.7604 mL
100 mM0.0276 mL0.1380 mL0.2760 mL1.3802 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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