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Tocainide
Catalog No. T13177LCas No. 41708-72-9
Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.
Tocainide
Catalog No. T13177LCas No. 41708-72-9
Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $38 | In Stock | |
| 25 mg | $63 | In Stock | |
| 50 mg | $92 | In Stock | |
| 100 mg | $137 | In Stock | |
| 200 mg | $198 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $29 | In Stock |
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Purity:99.84%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus. |
| Targets&IC50 | Na+ channel: |
| In vivo | Ventricular ectopic activity in unanesthetized dogs with coronary occlusion effectively suppressed by Tocainide (100 mg/kg). In both digitalis toxicity and coronary occlusion models, the Termination of tocainide infusion results in the prompt return of ventricular ectopic activity [1]. |
| Molecular Weight | 192.26 |
| Formula | C11H16N2O |
| Cas No. | 41708-72-9 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 11 mg/mL (57.21 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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