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LAU159

Catalog No. T11822 CAS 2055050-87-6

Purity 98.65% Datasheet

LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).

LAU159, CAS 2055050-87-6

Pack Size	Availability	Price/USD
1 mg	In stock	133.00
5 mg	In stock	271.00
10 mg	In stock	489.00
25 mg	In stock	701.00

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Purity 98.65%

HNMR HPLC COA Datasheet

Biological Description

Chemical Properties

Storage & Solubility Information

Description	LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
Targets&IC50	α1β3 GABA :ic50 （EC50）2.2 μM,

Molecular Weight	325.75
Formula	C17H12ClN3O2
CAS No.	2055050-87-6

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Varagic Z, et al. Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface. Br J Pharmacol. 2013 May;169(2):371-83.

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Answers to questions you may have can be found in the Inhibitor Handling Instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.