Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

SB-277011

Catalog No. T12861Cas No. 215803-78-4
Alias SB-277011A

SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.

SB-277011

SB-277011

Purity: 98.61%
Catalog No. T12861Alias SB-277011ACas No. 215803-78-4
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
Pack SizePriceAvailabilityQuantity
1 mg$39In Stock
5 mg$53In Stock
10 mg$85In Stock
25 mg$160In Stock
50 mg$267In Stock
100 mgInquiryIn Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "SB-277011"

Select Batch
Purity:98.61%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
Targets&IC50
5-HT1B:<5.2 (pKi), D2 receptor:6.0 (pKi), 5-HT1D:5.0 (pKi), D3 receptor:8.0 (pKi)
AliasSB-277011A
Chemical Properties
Molecular Weight438.56
FormulaC28H30N4O
Cas No.215803-78-4
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 4.39 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2802 mL11.4009 mL22.8019 mL114.0095 mL
5 mM0.4560 mL2.2802 mL4.5604 mL22.8019 mL
10 mM0.2280 mL1.1401 mL2.2802 mL11.4009 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy SB-277011 | purchase SB-277011 | SB-277011 cost | order SB-277011 | SB-277011 chemical structure | SB-277011 formula | SB-277011 molecular weight