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SB-277011

Catalog No. T12861Cas No. 215803-78-4
Alias SB-277011A

SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.

SB-277011

SB-277011

Purity: 98.61%
Catalog No. T12861Alias SB-277011ACas No. 215803-78-4
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
Pack SizePriceAvailabilityQuantity
1 mg$39In Stock
5 mg$53In Stock
10 mg$85In Stock
25 mg$160In Stock
50 mg$267In Stock
100 mgInquiryIn Stock
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Purity:98.61%
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Product Introduction

Bioactivity
Description
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
Targets&IC50
5-HT1D:5.0 (pKi), 5-HT1B:<5.2 (pKi), D2 receptor:6.0 (pKi), D3 receptor:8.0 (pKi)
AliasSB-277011A
Chemical Properties
Molecular Weight438.56
FormulaC28H30N4O
Cas No.215803-78-4
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 4.39 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2802 mL11.4009 mL22.8019 mL114.0095 mL
5 mM0.4560 mL2.2802 mL4.5604 mL22.8019 mL
10 mM0.2280 mL1.1401 mL2.2802 mL11.4009 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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