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VU 0255035

VU 0255035
VU 0255035 is a highly selective, competitive, and brain-penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM, used to reduce pilocarpine-induced seizures in mice and to examine the role of the M1 receptor in diverse situations.
Catalog No. T23508Cas No. 1135243-19-4
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Purity:98.26%
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VU 0255035

Catalog No. T23508Cas No. 1135243-19-4

VU 0255035 is a highly selective, competitive, and brain-penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM, used to reduce pilocarpine-induced seizures in mice and to examine the role of the M1 receptor in diverse situations.
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Pack SizePriceAvailabilityQuantity
5 mg$43In Stock
10 mg$73In Stock
25 mg$155In Stock
50 mg$232In Stock
100 mg$340In Stock
200 mg$475In Stock
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Product Introduction

Bioactivity
Description
VU 0255035 is a highly selective, competitive, and brain-penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM, used to reduce pilocarpine-induced seizures in mice and to examine the role of the M1 receptor in diverse situations.
Targets&IC50
M1 mACh:130 nM
Chemical Properties
Molecular Weight432.52
FormulaC18H20N6O3S2
Cas No.1135243-19-4
Storage & Solubility Information
Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 4.32 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.3120 mL11.5602 mL23.1203 mL115.6016 mL
5 mM0.4624 mL2.3120 mL4.6241 mL23.1203 mL
10 mM0.2312 mL1.1560 mL2.3120 mL11.5602 mL

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