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BAY 1892005
🥰Excellent
Catalog No. T77768Cas No. 2036352-13-1
BAY 1892005 is a p53 protein modulator that targets the p53 condenser for the study of diseases associated with misfolded p53 protein
BAY 1892005
🥰Excellent
Purity: 99.62%
Catalog No. T77768Cas No. 2036352-13-1
BAY 1892005 is a p53 protein modulator that targets the p53 condenser for the study of diseases associated with misfolded p53 protein
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $93 | In Stock | |
| 5 mg | $228 | In Stock | |
| 10 mg | $372 | In Stock | |
| 25 mg | $613 | In Stock | |
| 50 mg | $869 | In Stock | |
| 100 mg | $1,170 | In Stock | |
| 500 mg | $2,330 | In Stock |
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Purity:99.62%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | BAY 1892005 is a p53 protein modulator that targets the p53 condenser for the study of diseases associated with misfolded p53 protein |
| Targets&IC50 | p53-mutant:11.2 μM, H358:11.1 μM |
| In vitro | In p53-mutant cell lines Huh7 (IC50=11.2 μM) and H358 (IC50=11.1 μM), BAY 1892005 inhibits cell proliferation[1]. |
| Molecular Weight | 270.71 |
| Formula | C11H8ClFN2OS |
| Cas No. | 2036352-13-1 |
| Smiles | O=C(NC1=NC(=CS1)C=2C=CC=CC2F)CCl |
| Relative Density. | 1.454 g/cm3 at 20℃ (Predicted) |
Storage & Solubility Information
| Storage | store at low temperature | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 65 mg/mL (240.11 mM), Sonication is recommended.  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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