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CGP52432
🥰Excellent
Catalog No. T4363Cas No. 139667-74-6
Alias CGP 52432
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
CGP52432
🥰Excellent
Purity: 99.16%
Catalog No. T4363Alias CGP 52432Cas No. 139667-74-6
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $34 | In Stock | |
| 5 mg | $79 | In Stock | |
| 10 mg | $143 | In Stock | |
| 25 mg | $268 | In Stock | |
| 50 mg | $393 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $88 | In Stock |
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CitedSelect Batch
Purity:99.16%
Contact us for more batch information
With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM). |
| Targets&IC50 | GABAB:85 nM |
| Kinase Assay | Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000). |
| Alias | CGP 52432 |
| Molecular Weight | 384.24 |
| Formula | C15H24Cl2NO4P |
| Cas No. | 139667-74-6 |
| Smiles | C(NCCCP(C(OCC)OCC)(=O)O)C1=CC(Cl)=C(Cl)C=C1 |
| Relative Density. | 1.258 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 5 mg/mL (13.01 mM), Sonication and heating are recommended. | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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