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GSK 789472 hydrochloride
🥰Excellent
Catalog No. T22817Cas No. 1257326-24-1
Alias GSK-789472 HCl, 4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one, 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride
GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
GSK 789472 hydrochloride
🥰Excellent
Purity: 99.95%
Catalog No. T22817Alias GSK-789472 HCl, 4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one, 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochlorideCas No. 1257326-24-1
GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $37 | In Stock | |
| 2 mg | $53 | In Stock | |
| 5 mg | $88 | In Stock | |
| 10 mg | $133 | In Stock | |
| 25 mg | $268 | In Stock | |
| 50 mg | $392 | In Stock | |
| 100 mg | $592 | In Stock | |
| 200 mg | $783 | In Stock |
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CitedSelect Batch
Purity:99.95%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist. |
| Alias | GSK-789472 HCl, 4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one, 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride |
| Molecular Weight | 295.81 |
| Formula | C15H22ClN3O |
| Cas No. | 1257326-24-1 |
| Smiles | Cl.O=C1N(CC2CCCCN2)CCN1c1ccccc1 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 7.86 mg/mL (26.56 mM)  H2O: < 30 mg/mL (101.42 mM) | ||||||||||||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||||||||||||
DMSO/H2O
H2O
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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