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Indinavir sulfate
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Indinavir sulfate
Catalog No. T5863Cas No. 157810-81-6
Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $139 | In Stock | |
| 50 mg | $198 | In Stock | |
| 100 mg | $298 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $58 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM. |
| In vitro | At low concentrations (0.0003-10?μmol/l) indinavir acts as a positive allosteric modulator (EC50?=?0.021?μmol/l), whereas at concentrations greater than 10?μmol/l (30-100?μmol/l) indinavir acts as an inhibitor of the α7-nicotinic acetylcholine receptor. |
| Alias | L735524 sulfate, MK-639 sulfate |
| Molecular Weight | 711.87 |
| Formula | C36H49N5O8S |
| Cas No. | 157810-81-6 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 100 mg/mL (140.48 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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Keywords
InhibitorMK639L-735524 SulfateL 735524Huh7Matrix metalloproteinasesL-735524PBMCMK 639Indinavir sulfateMMPMK-639Indinavir SulfateSARS coronavirusHIV ProteaseApoptosishepatocarcinomasL735524L735524 SulfateHuman immunodeficiency virusMK-639 SulfateIndinavirinhibitCD4 T cellsMK639 SulfateMK 639 SulfateHIVL 735524 SulfateSARS-CoV
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