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PD 168568 dihydrochloride
🥰Excellent
Catalog No. T12383Cas No. 1782532-06-2
Alias PD 168568 (dihydrochloride)
PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
PD 168568 dihydrochloride
🥰Excellent
Purity: 99.27%
Catalog No. T12383Alias PD 168568 (dihydrochloride)Cas No. 1782532-06-2
PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $40 | In Stock | |
| 10 mg | $53 | In Stock | |
| 25 mg | $119 | In Stock | |
| 50 mg | $178 | In Stock | |
| 100 mg | $260 | In Stock | |
| 200 mg | $366 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $55 | In Stock |
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Purity:99.27%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM). |
| Targets&IC50 | D4 receptor:8.8 nM (ki) |
| In vitro | PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor)[1]. |
| In vivo | PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat[1]. |
| Alias | PD 168568 (dihydrochloride) |
| Molecular Weight | 422.39 |
| Formula | C22H29Cl2N3O |
| Cas No. | 1782532-06-2 |
| Smiles | O=C1NC(CCN2CCN(CC2)C3=CC=C(C)C(C)=C3)C4=C1C=CC=C4.Cl.Cl |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 55 mg/mL (130.21 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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