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TC-2216
🥰Excellent
Catalog No. T68154Cas No. 646055-67-6
TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.
TC-2216
🥰Excellent
Purity: 100.00%
Catalog No. T68154Cas No. 646055-67-6
TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $86 | In Stock | |
| 5 mg | $200 | In Stock | |
| 10 mg | $300 | In Stock | |
| 25 mg | $586 | In Stock | |
| 50 mg | $800 | In Stock | |
| 100 mg | $1,090 | In Stock | |
| 500 mg | $2,230 | In Stock |
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CitedSelect Batch
Purity:100.00%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression. |
| Targets&IC50 | α4β2 nAChR:0.042 µM(Ki), α4β2 nAChR:0.901 µM, α7 nAChR:6.9 µM(Ki) |
| In vitro | TC-2216 (6.0-133 mL/tree; injected) alleviate the rapid spread of tree wilt disease.[3] |
| Molecular Weight | 203.28 |
| Formula | C12H17N3 |
| Cas No. | 646055-67-6 |
| Smiles | C12(CN(CC1)C=3C=CC=NC3)CCCN2 |
Storage & Solubility Information
| Storage | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (245.97 mM), Sonication is recommended.  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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