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Tetrabenazine Racemate
😃Good
Catalog No. T3534Cas No. 718635-93-9
Alias TETRABENAZINE, Rubigen, Ro 1-9569 Racemate, Nitoman
Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affinity label for the vesicle transport system.
Tetrabenazine Racemate
😃Good
Purity: 98.86%
Catalog No. T3534Alias TETRABENAZINE, Rubigen, Ro 1-9569 Racemate, NitomanCas No. 718635-93-9
Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affinity label for the vesicle transport system.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $46 | In Stock | |
| 25 mg | $83 | In Stock | |
| 50 mg | $124 | In Stock | |
| 100 mg | $165 | In Stock | |
| 200 mg | $216 | Backorder |
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Purity:98.86%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affinity label for the vesicle transport system. |
| In vivo | BMS-663068 has good antiviral activity in subjects infected with virus shown to be susceptible (IC50, <100 nM) to the agent[1]. |
| Alias | TETRABENAZINE, Rubigen, Ro 1-9569 Racemate, Nitoman |
| Molecular Weight | 317.42 |
| Formula | C19H27NO3 |
| Cas No. | 718635-93-9 |
| Smiles | COc1cc2CCN3CC(CC(C)C)C(=O)CC3c2cc1OC |
| Relative Density. | 1.12 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 55 mg/mL (173.27 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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