Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor. PNU-177864 hydrochloride is structurally consistent with a cationic amphiphilic drug (CAD). PNU-177864 hydrochloride induces phospholipidosis in vivo. PNU-177864 hydrochloride exhibits antischizophrenic activity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 50.00 | |
10 mg | In stock | $ 75.00 | |
25 mg | In stock | $ 128.00 | |
50 mg | In stock | $ 192.00 | |
100 mg | In stock | $ 287.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 73.00 |
Description | PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor. PNU-177864 hydrochloride is structurally consistent with a cationic amphiphilic drug (CAD). PNU-177864 hydrochloride induces phospholipidosis in vivo. PNU-177864 hydrochloride exhibits antischizophrenic activity. |
In vivo | In Sprague-Dawley rats, PNU-177864 hydrochloride (8-200 mg/kg; gavage) induces phospholipidosis in unusual target organs including epididymis, hair follicles and pituitary[1]. |
Synonyms | PNU-177864 (hydrochloride) |
Molecular Weight | 438.89 |
Formula | C18H22ClF3N2O3S |
CAS No. | 1783978-03-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (113.92 mM)
You can also refer to dose conversion for different animals. More
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PNU-177864 hydrochloride 1783978-03-9 GPCR/G Protein Neuroscience Dopamine Receptor PNU 177864 Hydrochloride PNU-177864 Hydrochloride PNU177864 PNU-177864 PNU177864 Hydrochloride PNU-177864 (hydrochloride) PNU 177864 inhibitor inhibit