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Benzbromarone
🥰Excellent
Catalog No. T1274Cas No. 3562-84-3
Alias Urinorm, Normurat, Desuric
Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.
Benzbromarone
🥰Excellent
Purity: 100%
Catalog No. T1274Alias Urinorm, Normurat, DesuricCas No. 3562-84-3
Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 50 mg | $33 | In Stock | |
| 100 mg | $47 | In Stock | |
| 200 mg | $60 | In Stock | |
| 500 mg | $95 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $47 | In Stock |
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Purity:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM. |
| Targets&IC50 | CYP2C9:19.3 nM(Ki) |
| In vivo | In oocytes expressing URAT1 (IC50 <0.1 μM), Benzbromarone (50 μM) completely inhibited the uptake of uric acid. In rat hepatocytes, Benzbromarone (100 μM) increased mitochondrial size and induced apoptosis in 11% of cells. |
| Alias | Urinorm, Normurat, Desuric |
| Molecular Weight | 424.08 |
| Formula | C17H12Br2O3 |
| Cas No. | 3562-84-3 |
| Smiles | C(=O)(C=1C=2C(OC1CC)=CC=CC2)C3=CC(Br)=C(O)C(Br)=C3 |
| Relative Density. | 1.709 g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
| Solubility Information | Ethanol: 9 mg/mL (21.22 mM) DMSO: 70 mg/mL (165.06 mM)  H2O: < 1 mg/mL (insoluble or slightly soluble) | ||||||||||||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||||||||||||
Ethanol/DMSO
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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