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GR 103691
GR 103691, a potent and selective dopamine D3 receptor antagonist (Ki: 0.4 nM), exhibits more than 100-fold selectivity for human dopamine D3 receptors over human D4 and D1 sites.
Catalog No. T11463Cas No. 162408-66-4
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Purity:99.29%
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GR 103691
Catalog No. T11463Cas No. 162408-66-4
GR 103691, a potent and selective dopamine D3 receptor antagonist (Ki: 0.4 nM), exhibits more than 100-fold selectivity for human dopamine D3 receptors over human D4 and D1 sites.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $38 | In Stock | |
| 5 mg | $61 | In Stock | |
| 10 mg | $101 | In Stock | |
| 25 mg | $207 | In Stock | |
| 50 mg | $328 | In Stock | |
| 100 mg | $531 | In Stock | |
| 500 mg | $1,180 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | GR 103691, a potent and selective dopamine D3 receptor antagonist (Ki: 0.4 nM), exhibits more than 100-fold selectivity for human dopamine D3 receptors over human D4 and D1 sites. |
| Targets&IC50 | D3:ki:0.4 nM |
| In vitro | GR 103691 shows a marked affinity for α-1 adrenoceptors (Ki: 12.6 nM) and serotonin1A (5-HT1A) receptors (Ki: 5.8 nM). |
| Molecular Weight | 485.62 |
| Formula | C30H35N3O3 |
| Cas No. | 162408-66-4 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 4.86 mg/mL (10 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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