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Nelfinavir Mesylate

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Purity:98.27%

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COA HPLC HNMR

Nelfinavir Mesylate

Catalog No. T6001Cas No. 159989-65-8

Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).

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Pack Size	Price	Availability
5 mg	$48	In Stock
10 mg	$74	In Stock
25 mg	$157	In Stock
50 mg	$266	In Stock
100 mg	$397	In Stock
1 mL x 10 mM (in DMSO)	$72	In Stock

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Product Introduction

Bioactivity

Description	Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).
Kinase Assay	GTPγ[35S] binding assay: The cells are homogenized and centrifuged at 26900 × g for 30 min at 4°C. Membranes are re-suspended in 20 mM HEPES (pH 7.4), 100 mM NaCl, 10 mM MgCl2, 1 mM EDTA and 0.1% fat-free BSA at 2–3 mg protein/mL. GTPγ[35S] binding assay is performed with the membranes (75 mg protein /mL in 50 mM HEPES, 100 mM NaCl, 10 mM MgCl2, 20 μg/mL saponin and 0.1% fat-free BSA (pH 7.4), 5 mg/mL with wheat-germ agglutinin-coated scintillation proximity assay-bead, and 10 μM GDP for 10–15 min. The GTPγ[35S]-binding reaction is started by the addition of 200 pM GTPγ[35S]. After 120 min at room temperature, the plates are centrifuged for 10 min at 300 × g and counted.
Alias	Viracept, Nelfin, AG1343, AG 1343 Mesylate

Chemical Properties

Molecular Weight	663.89
Formula	C33H49N3O7S2
Cas No.	159989-65-8

Storage & Solubility Information

Storage

keep away from direct sunlight,store at low temperature Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: < 1 mg/mL (insoluble or slightly soluble)

DMSO: 93 mg/mL (140.1 mM)

Ethanol: 93 mg/mL (140.1 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.5063 mL	7.5314 mL	15.0627 mL	75.3137 mL
5 mM	0.3013 mL	1.5063 mL	3.0125 mL	15.0627 mL
10 mM	0.1506 mL	0.7531 mL	1.5063 mL	7.5314 mL
20 mM	0.0753 mL	0.3766 mL	0.7531 mL	3.7657 mL
50 mM	0.0301 mL	0.1506 mL	0.3013 mL	1.5063 mL
100 mM	0.0151 mL	0.0753 mL	0.1506 mL	0.7531 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc