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Tolterodine
Catalog No. T23229Cas No. 124937-51-5
Alias PNU-200583, (R)-Tolterodine, (R)-(+)-Tolterodine, (+)-Tolterodine
Tolterodine ((R)-(+)-Tolterodine) is a novel and selective muscarinic-type receptor (mAChR) antagonist used in the treatment of detrusor instability and overactive bladder syndrome.
Tolterodine
Catalog No. T23229Alias PNU-200583, (R)-Tolterodine, (R)-(+)-Tolterodine, (+)-TolterodineCas No. 124937-51-5
Tolterodine ((R)-(+)-Tolterodine) is a novel and selective muscarinic-type receptor (mAChR) antagonist used in the treatment of detrusor instability and overactive bladder syndrome.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $30 | In Stock | |
| 10 mg | $36 | In Stock | |
| 25 mg | $56 | In Stock | |
| 50 mg | $80 | In Stock |
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Purity:99.71%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tolterodine ((R)-(+)-Tolterodine) is a novel and selective muscarinic-type receptor (mAChR) antagonist used in the treatment of detrusor instability and overactive bladder syndrome. |
| In vivo | Tolterodine, as a competitive muscarinic acetylcholine receptor antagonist, works by binding to muscarinic receptors, preventing acetylcholine from binding to its receptors, thereby reducing the contractions of the bladder smooth muscle. |
| Alias | PNU-200583, (R)-Tolterodine, (R)-(+)-Tolterodine, (+)-Tolterodine |
| Molecular Weight | 325.49 |
| Formula | C22H31NO |
| Cas No. | 124937-51-5 |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (245.78 mM), Sonication is recommended. Ethanol: 100 mg/mL (307.23 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO/Ethanol
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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