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5-HT2 antagonist 1
🥰Excellent
Catalog No. T12597Cas No. 191592-09-3
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist with weak α1 adrenoceptor blocking activity.
5-HT2 antagonist 1
🥰Excellent
Purity: 99.25%
Catalog No. T12597Cas No. 191592-09-3
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist with weak α1 adrenoceptor blocking activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $714 | In Stock | |
| 5 mg | $1,430 | In Stock | |
| 10 mg | $1,930 | In Stock | |
| 25 mg | $2,870 | In Stock | |
| 50 mg | $3,870 | In Stock | |
| 100 mg | $5,230 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $1,690 | In Stock |
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CitedSelect Batch
Purity:99.25%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | 5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist with weak α1 adrenoceptor blocking activity. |
| In vitro | 5-HT2 antagonist 1 displays dose-dependent inhibition of serotonin (erotonin)-induced contraction in guinea pig mesenteric artery, exhibiting 45%, 88%, and 93% inhibition at concentrations of 10 nM, 100 nM, and 1000 nM, respectively. Conversely, it demonstrates minimal inhibition of norepinephrine-induced contraction in guinea pig aorta, with 1% and 10% inhibition at 10 nM and 100 nM, respectively[1]. |
| Molecular Weight | 400.49 |
| Formula | C22H29FN4O2 |
| Cas No. | 191592-09-3 |
| Smiles | CN1C2=C(C(=O)N(CCCN3CCN(CC3)C4=CC=C(F)C=C4)CCC2O)C=C1 |
| Relative Density. | 1.28 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 45 mg/mL (112.36 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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