Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 34.00 | |
2 mg | In stock | $ 48.00 | |
5 mg | In stock | $ 77.00 | |
10 mg | In stock | $ 116.00 | |
25 mg | In stock | $ 195.00 | |
50 mg | In stock | $ 288.00 | |
100 mg | In stock | $ 433.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 88.00 |
Description | Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. |
Targets&IC50 | 5-HT2:0.9 nM, α2-adrenoceptor:150 nM, D2:70 nM, α1-adrenoceptor:97 nM, H1:35 nM |
In vitro | Ritanserin less active on Histamine-H1 (IC50, 35 nM), Dopamine-D2 (IC50, 70 nM), Adrenergic-α1 (IC50, 97 nM), Adrenergic-α2 receptor (IC50, 150 nM) [1]. |
Synonyms | R 55667 |
Molecular Weight | 477.57 |
Formula | C27H25F2N3OS |
CAS No. | 87051-43-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (52.35 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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Ritanserin 87051-43-2 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor Adrenergic Receptor 5-HT Receptor Dopamine Receptor Inhibitor 5-hydroxytryptamine Receptor inhibit Serotonin Receptor R-55667 R55667 Beta Receptor R 55667 inhibitor