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GR 125743

🥰Excellent
Catalog No. T8737Cas No. 148547-33-5

GR 125743 is a novel antagonist of 5-HT1B/1D receptor.

GR 125743

GR 125743

🥰Excellent
Purity: 99.76%
Catalog No. T8737Cas No. 148547-33-5
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
Pack SizePriceAvailabilityQuantity
1 mg$36In Stock
2 mg$51In Stock
5 mg$80In Stock
10 mg$122In Stock
25 mg$247In Stock
50 mg$369In Stock
100 mg$549In Stock
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Purity:99.76%
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Product Introduction

Bioactivity
Description
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
In vitro
GR-125743, a new radiolabelled derivative of a compound that exhibits selective antagonistic properties with respect to the serotonin human (h5-HT1D) and human (h5-HT1B) receptors.?The compound has been characterized for its ability to label the cloned h5-HT1D and h5-HT1B receptors.
Chemical Properties
Molecular Weight416.52
FormulaC25H28N4O2
Cas No.148547-33-5
SmilesCOc1ccc(NC(=O)c2ccc(c(C)c2)-c2ccncc2)cc1N1CCN(C)CC1
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 4.17 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4008 mL12.0042 mL24.0085 mL120.0423 mL
5 mM0.4802 mL2.4008 mL4.8017 mL24.0085 mL
10 mM0.2401 mL1.2004 mL2.4008 mL12.0042 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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