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Azaphen

Catalog No. T7521 CAS 24853-80-3

Synonyms: Pipofezine hydrochloride, Pipofezin hydrochloride, Pipofezin, inhibit, Inhibitor, Pipofezine, Serotonin Transporter, Azaphen, SERT, 5-HTT, SLC6A4, Azafen

Azaphen is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.

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Azaphen, CAS 24853-80-3

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Azaphen is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.

Synonyms	Pipofezine hydrochloride, Pipofezin hydrochloride, Pipofezin, inhibit, Inhibitor, Pipofezine, Serotonin Transporter, Azaphen, SERT, 5-HTT, SLC6A4, Azafen
Molecular Weight	370.28
Formula	C16H21Cl2N5O
CAS No.	24853-80-3

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: Insoluble

H2O: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Aleeva G N , Molodavkin G M , Voronina T A . Comparison of Antidepressant Effects of Azafan, Tianeptine, and Paroxetine[J]. Bull Exp Biol Med, 2009, 148(1):54-56.

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Neurotransmitter Receptor Compound Library Inhibitor Library Neuronal Signaling Compound Library Anti-Neurodegenerative Disease Compound Library Bioactive Compound Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.