Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 179.00 | |
5 mg | In stock | $ 455.00 | |
10 mg | In stock | $ 672.00 | |
25 mg | In stock | $ 1,060.00 | |
50 mg | In stock | $ 1,430.00 | |
100 mg | In stock | $ 1,920.00 | |
500 mg | In stock | $ 3,850.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 490.00 |
Description | Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors. |
Molecular Weight | 399.36 |
Formula | C19H28Cl2N4O |
CAS No. | 839712-25-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10.2 mg/mL (25.6 mM), ultrasonic and warming and heat to 80°C
You can also refer to dose conversion for different animals. More
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Didesmethyl cariprazine 839712-25-3 GPCR/G Protein Neuroscience Dopamine Receptor 5-HT Receptor inhibitor inhibit