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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $97 | In Stock | |
5 mg | $239 | In Stock | |
10 mg | $378 | In Stock | |
25 mg | $687 | In Stock | |
50 mg | $977 | In Stock | |
100 mg | $1,360 | In Stock | |
500 mg | $2,730 | In Stock | |
1 mL x 10 mM (in DMSO) | $263 | In Stock |
Description | Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM). It is development as an injectable agent for the treatment of postoperative pain. |
Targets&IC50 | 5-HT2A receptor:1.3 μM, GlyT2:0.86 μM, P2X3 (rat):0.87 μM |
Molecular Weight | 430.97 |
Formula | C21H35ClN2O5 |
Cas No. | 1440796-75-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 50 mg/mL (116.02 mM) ![]() | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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