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Cerlapirdine
🥰Excellent
Catalog No. T30798Cas No. 925448-93-7
Alias WAY-262,531, SAM-531, SAM531, SAM 531, PF-05212365, PF05212365, P -05212365
Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
Cerlapirdine
🥰Excellent
Purity: 98.60%
Catalog No. T30798Alias WAY-262,531, SAM-531, SAM531, SAM 531, PF-05212365, PF05212365, P -05212365Cas No. 925448-93-7
Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $74 | In Stock | |
| 5 mg | $178 | In Stock | |
| 10 mg | $289 | In Stock | |
| 25 mg | $572 | In Stock | |
| 50 mg | $822 | In Stock | |
| 100 mg | $1,130 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $209 | In Stock |
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CitedSelect Batch
Purity:98.60%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist. |
| Alias | WAY-262,531, SAM-531, SAM531, SAM 531, PF-05212365, PF05212365, P -05212365 |
| Molecular Weight | 409.5 |
| Formula | C22H23N3O3S |
| Cas No. | 925448-93-7 |
| Smiles | S(=O)(=O)(C=1C=2C(NN1)=CC=C(OCCCN(C)C)C2)C=3C4=C(C=CC3)C=CC=C4 |
| Relative Density. | 1.300 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 38 mg/mL (92.80 mM), when pH Adjusted to 3 with HCl. Sonication and heating to 60℃ are recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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