Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

Glycopyrrolate

Catalog No. T2387Cas No. 596-51-0
Alias Robinul, Glycopyrronium bromide, Glycopyrrolate bromide, Gastrodyn

Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.

Glycopyrrolate

Glycopyrrolate

Purity: 99.86%
Catalog No. T2387Alias Robinul, Glycopyrronium bromide, Glycopyrrolate bromide, GastrodynCas No. 596-51-0
Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.
Pack SizePriceAvailabilityQuantity
5 mg$32In Stock
10 mg$48In Stock
25 mg$58In Stock
50 mg$90In Stock
100 mg$130In Stock
500 mg$318In Stock
1 mL x 10 mM (in DMSO)$50In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "Glycopyrrolate"

Select Batch
Purity:99.86%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.
In vitro
Glycopyrrolate inhibits EFS-induced contraction of guinea-pig trachea and human airways in a concentration-dependent manner. In competition studies, glycopyrrolate binds human peripheral lung and human airway smooth muscle (HASM) muscarinic receptors with affinities in the nanomolar range (Ki values 0.5–3.6?nM). Glycopyrrolate showed no selectivity in its binding to the M1–M3 receptors. Kinetics studies show that glycopyrrolate dissociates slowly from HASM muscarinic receptors[1].
AliasRobinul, Glycopyrronium bromide, Glycopyrrolate bromide, Gastrodyn
Chemical Properties
Molecular Weight398.33
FormulaC19H28BrNO3
Cas No.596-51-0
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 50 mg/mL (125.52 mM), Sonication is recommended.
H2O: 72 mg/mL (180.8 mM)
Ethanol: 55 mg/mL (138.1 mM)
Solution Preparation Table
DMSO/Ethanol/H2O
1mg5mg10mg50mg
1 mM2.5105 mL12.5524 mL25.1048 mL125.5241 mL
5 mM0.5021 mL2.5105 mL5.0210 mL25.1048 mL
10 mM0.2510 mL1.2552 mL2.5105 mL12.5524 mL
20 mM0.1255 mL0.6276 mL1.2552 mL6.2762 mL
50 mM0.0502 mL0.2510 mL0.5021 mL2.5105 mL
100 mM0.0251 mL0.1255 mL0.2510 mL1.2552 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy Glycopyrrolate | purchase Glycopyrrolate | Glycopyrrolate cost | order Glycopyrrolate | Glycopyrrolate chemical structure | Glycopyrrolate in vitro | Glycopyrrolate formula | Glycopyrrolate molecular weight