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Alizapride hydrochloride

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Purity:99.71%

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COA HNMR HPLC

Alizapride hydrochloride

Catalog No. T2574Cas No. 59338-87-3

Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.

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Pack Size	Price	Availability
25 mg	$48	In Stock
50 mg	$71	In Stock
100 mg	$113	In Stock
200 mg	$168	In Stock
500 mg	$283	In Stock
1 mL x 10 mM (in DMSO)	$39	In Stock

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Product Introduction

Bioactivity

Description	Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.
In vitro	Intravenous administration of 5 mg/kg Alizapride in rats effectively counteracts the reduction in gastrointestinal motility induced by the given dose of Apomorphine. Alizapride exhibits low toxicity in mice and rats, particularly when administered extragastrically. Following oral or extragastric administration, Alizapride is primarily excreted in its unmodified form; however, approximately 25% of Alizapride undergoes metabolic transformation before excretion.
In vivo	Alizapride contains an N-allyl moiety, which may undergo N-deallylation and/or epoxidation, potentially leading to the formation of chemically reactive metabolites.
Alias	Alizapride HCl

Chemical Properties

Molecular Weight	351.83
Formula	C16H21N5O2·HCl
Cas No.	59338-87-3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 50 mg/mL (142.11 mM)

Ethanol: < 1 mg/mL (insoluble or slightly soluble)

DMSO: 40 mg/mL (113.69 mM)

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	2.8423 mL	14.2114 mL	28.4228 mL	142.1141 mL
5 mM	0.5685 mL	2.8423 mL	5.6846 mL	28.4228 mL
10 mM	0.2842 mL	1.4211 mL	2.8423 mL	14.2114 mL
20 mM	0.1421 mL	0.7106 mL	1.4211 mL	7.1057 mL
50 mM	0.0568 mL	0.2842 mL	0.5685 mL	2.8423 mL
100 mM	0.0284 mL	0.1421 mL	0.2842 mL	1.4211 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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