Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

Azacyclonol

🥰Excellent
Catalog No. T0318Cas No. 115-46-8
Alias γ-pipradol, MER 17, MDL 4829, Ataractan

Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.

Azacyclonol

Azacyclonol

🥰Excellent
Purity: 99.61%
Catalog No. T0318Alias γ-pipradol, MER 17, MDL 4829, AtaractanCas No. 115-46-8
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
Pack SizePriceAvailabilityQuantity
1 g$29In Stock
1 mL x 10 mM (in DMSO)$29In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "Azacyclonol"

Select Batch
Purity:99.61%
Contact us for more batch information
Resource Download
With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.

Product Introduction

Bioactivity
Description
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
In vitro
Azacyclonol exhibits an inhibitory effect on the activity of feline cervical sympathetic ganglia by 6.63%. Intravenous injection of Azacyclonol modifies the nictitating membrane's response to postganglionic and preganglionic stimulation.
In vivo
Azacyclonol affects human hepatic microsomes with apparent Km and Vmax values of 0.82 μM and 60 pmol/min/mg, respectively. In human intestinal microsomes, the formation of azacyclonol is time-dependent, demonstrating linearity up to 60 minutes. The rate of azacyclonol formation increases linearly with microsomal protein concentrations reaching 2 mg/mL.
Aliasγ-pipradol, MER 17, MDL 4829, Ataractan
Chemical Properties
Molecular Weight267.37
FormulaC18H21NO
Cas No.115-46-8
SmilesOC(C1CCNCC1)(C1=CC=CC=C1)C1=CC=CC=C1
Relative Density.Ca. 1.103 g/cm3.
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
Ethanol: 49 mg/mL (183.3 mM)
H2O: 2 mg/mL (7.48 mM)
DMSO: 50 mg/mL (187.01 mM)
Solution Preparation Table
H2O/Ethanol/DMSO
1mg5mg10mg50mg
1 mM3.7401 mL18.7007 mL37.4014 mL187.0068 mL
5 mM0.7480 mL3.7401 mL7.4803 mL37.4014 mL
Ethanol/DMSO
1mg5mg10mg50mg
10 mM0.3740 mL1.8701 mL3.7401 mL18.7007 mL
20 mM0.1870 mL0.9350 mL1.8701 mL9.3503 mL
50 mM0.0748 mL0.3740 mL0.7480 mL3.7401 mL
100 mM0.0374 mL0.1870 mL0.3740 mL1.8701 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy Azacyclonol | purchase Azacyclonol | Azacyclonol cost | order Azacyclonol | Azacyclonol chemical structure | Azacyclonol in vivo | Azacyclonol in vitro | Azacyclonol formula | Azacyclonol molecular weight