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Pimethixene
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Purity:99.1%
Pimethixene
Catalog No. T12489Cas No. 314-03-4
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $35 | In Stock | |
| 2 mg | $48 | In Stock | |
| 5 mg | $71 | In Stock | |
| 10 mg | $101 | In Stock | |
| 25 mg | $180 | In Stock | |
| 50 mg | $267 | In Stock | |
| 100 mg | $397 | In Stock | |
| 200 mg | $593 | In Stock | |
| 500 mg | $949 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $81 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively). |
| Targets&IC50 | 5-HT2A receptor:10.22 (pki), 5-HT2C receptor:8.42 (pki), H1 receptor:10.14 (pki), D2 receptor:8.19 (pki), M1 receptor:8.61 (pki), 5-HT1A receptor:7.63 (pki), DD4.4 receptor:7.54 (pki), M2 mAChR:9.38 (pki), 5-HT2B receptor:10.44 (pki) |
| Alias | Calmixen, Pimetixene |
| Molecular Weight | 293.43 |
| Formula | C19H19NS |
| Cas No. | 314-03-4 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 18.33 mg/ml (62.48 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
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