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Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $30 | In Stock | |
10 mg | $48 | In Stock | |
25 mg | $77 | In Stock | |
50 mg | Inquiry | In Stock | |
1 mL x 10 mM (in DMSO) | $53 | In Stock |
Description | Pimethixene maleate (Pimetixene maleate) is a potent 5-HT2B receptor antagonist with sedative and antitussive activity.Pimethixene maleate inhibits 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2, and can be used in studies of dry and irritant cough in children. irritant cough in children. |
Targets&IC50 | H1 receptor:10.14 (pKi), 5-HT2B receptor:10.44 (pKi), DD4.4 receptor:7.54 (pKi), 5-HT2A receptor:10.22 (pKi), M1 receptor:8.61 (pKi), D2 receptor:8.19 (pKi), M2 mAChR:9.38 (pKi), 5-HT2C receptor:8.42 (pKi), 5-HT1A receptor:7.63 (pKi) |
Alias | Pimetixene maleate |
Molecular Weight | 409.5 |
Formula | C23H23NO4S |
Cas No. | 13187-06-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 80 mg/mL (195.36 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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