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Eltoprazine hydrochloride
🥰Excellent
Catalog No. T7498Cas No. 98206-09-8
Alias DU 28853 hydrochloride
Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively).
Eltoprazine hydrochloride
🥰Excellent
Purity: 99.94%
Catalog No. T7498Alias DU 28853 hydrochlorideCas No. 98206-09-8
Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $40 | In Stock | |
| 10 mg | $73 | In Stock | |
| 25 mg | $147 | In Stock | |
| 50 mg | $272 | In Stock | |
| 100 mg | $396 | In Stock | |
| 500 mg | $927 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $44 | In Stock |
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CitedSelect Batch
Purity:99.94%
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With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively). |
| Targets&IC50 | 5-HT2B:81 nM, 5-HT1B:52 nM , 5-HT1A:40 nM |
| In vivo | Eltoprazine hydrochloride exerts a dose-dependent decrease in aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg)[1]. |
| Alias | DU 28853 hydrochloride |
| Molecular Weight | 256.73 |
| Formula | C12H17ClN2O2 |
| Cas No. | 98206-09-8 |
| Smiles | Cl.c1cc2c(c(N3CCNCC3)c1)OCCO2 |
| Relative Density. | 1.18g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 31 mg/mL (120.75 mM) H2O: 28 mg/mL (109.06 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
H2O/DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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