Welcome to our new website experience

As we continue to roll out more enhancements, enjoy a host of updated features to make your journey with us smarter, faster and easier.

What's new

Intuitive search with relevant results
Easily compare products in detail
Quick, simple checkout
Be part of our community, read or submit product reviews

We would love to know what you think, so we have included a feedback tab on every page.

Popular Searches

Wikimole

1Trametinib
2Necrostatin-1
3Bortezomib
4LY294002
5Insulin (human)

New Product

1PALDA
2IACS-52825
3Brigimadlin
4Gimsilumab
5SB 216641 hydrochloride

Compound Library

1DNA Damage & Repair Compound Library
2GPCR Compound Library
3Anti-Nervous System Disease Library
4Stem Cell Differentiation Compound Library
5Anti-Cardiovascular Disease Compound Library

Home

All

Inhibitors & Agonists

Compound Libraries

Focused Bioactive Libraries
Natural Product Libraries
Fragment Libraries
Drug-like Compound Libraries
Natural Products
Recombinant Proteins
Technical Services
Popular product application
Reagent Kits
Biochemicals

Autophagy
Cell Cycle/Checkpoint
Cytoskeletal Signaling
Chromatin/Epigenetic
Endocrinology/Hormones
Hedgehog/Smoothened
Angiogenesis
DNA Damage/DNA Repair
Apoptosis
NF-κB
Neuroscience
MAPK
Microbiology/Virology
GPCR/G Protein
TGF-beta/Smad
Immunology/Inflammation
Proteases/Proteasome
Stem Cells
Ubiquitination
Oxidation-Reduction
Membrane transporter/Ion channel
PI3K/Akt/mTOR signaling
Metabolism
Wnt/beta-catenin
JAK/STAT signaling
Tyrosine Kinase/Adaptors
TLR
PARP
Antibody-drug Conjugate/ADC Related
Focused Bioactive Libraries Approved Drug Library FDA-Approved Drug Library FDA-Approved & Pharmacopeia Drug Library Clinical Compound Library Preclinical Compound Library Bioactive Compound Library Target-Focused Phenotypic Screening Library ReFRAME Related Library Epigenetics Compound Library Cytoskeletal Signaling Pathway Compound Library Transcription Factor-Targeted Compound Library GPCR Compound Library Ion Channel Inhibitor Library Endocrinology-Hormone Compound Library JAK-STAT Compound Library NF-κB Signaling Compound Library DNA Damage & Repair Compound Library Ubiquitination Compound Library Ferroptosis Compound Library Cuproptosis Compound Library Kinase Inhibitor Library Anti-Cancer Compound Library Anti-Bacterial Compound Library Anti-Cardiovascular Disease Compound Library CNS-Penetrant Compound Library Anti-Viral Compound Library Anti-Neurodegenerative Disease Compound Library Peptide Compound Library
Natural Product Libraries Natural Product Library for HTS Natural Product Library Human Endogenous Metabolite Library Human Endogenous Metabolite Compound Library Plus Natural Product Derivatives Library Polyphenolic Natural Product Library Alkaloid Natural Product Library Flavonoid Natural Product Library Terpene Natural Product Library Covalent Natural Product Library The Yao nationality medicine Library Tibetan medicine Compound Library Traditional Mongolian Medicine Compound Library Food as Medicine Compound Library Marine Natural Product Library Microbial Natural Product Library Anti-infective Natural Product Library Anti-Tumor Natural Product Library Anti-Inflammatory Traditional Chinese Medicine Compound Library Anti-COVID-19 Traditional Chinese Medicine Compound Library Anti-virus Traditional Chinese Medicine Monomer Library Anti-Colorectal Cancer Traditional Chinese Medicine Compound Library PBCRBS Traditional Chinese Medicine Compound Library Traditional Chinese Medicine Monomer Library Selected Plant-Sourced Compound Library Gut Microbial Metabolite Library Selectable Natural Product Library Natural Product Derivatives Library for CADD
Fragment Libraries High Solubility Fragment Library Drug-Fragment Library
Drug-like Compound Libraries Mini Scaffold Library Golden Scaffold Library SmartTM Library Diversity Core Library Part1 Covalent Inhibitor Library Drug-like natural compound library
Steroids
Coumarins
Lignans
Saccharides and Glycosides
Alkaloids
Terpenoids
Phenylpropanoids
Flavonoids
Phenols
Quinones
Others
CAR-T Therapy Target Proteins
CD Proteins
Complement System
Cytokines and Growth Factors
Enzymes
Fluorescent Proteins
Hormones
Immune Checkpoint Proteins
Others
Receptor Proteins
Viral Proteins
Molecular Docking
Virtual Screening
Biomolecular Interaction
Custom Synthesis
AI-driven Ultra High-throughput Virtual Screening
Tumor/Cancer
Immune and Inflammatory
Neurodegenerative Diseases
Endocrine and Metabolism
Cardiovascular Diseases
Infectious Diseases
Organoids and Stem Cells
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktail
Protease Inhibitor Cocktail
Phosphatase Inhibitor Cocktail
Deacetylase Inhibitor Cocktail
RIPA Lysis Buffer
BCA Protein Quantification Kit
Sterile Antibiotic Solution
Magnetic Beads
Immunoprecipitation Beads
Immunoprecipitation Kits
Streptavidin Magnetic Beads
Protein Purification Magnetic Beads
Cell Isolation Kits
Preactivated Magnetic Beads
Polymer Magnetic Beads
Agarose Magnetic Beads
Dextran Magnetic Beads
Agarose Beads
Inhibitory Antibodies
Peptides
PROTAC
E3 Ligase Ligand-Linker Conjugate
Ligand for E3 Ligase
Ligand for Target Protein for PROTAC
Linker
PROTAC Selection
PROTAC-linker Conjugate for PAC
SNIPER
Target Protein Ligand-Linker Conjugate
dyes
Isotope products
Deuterium Labeled Compounds
Carbon-13 Labeled Compounds
Nitrogen-15 Labeled Compounds
Antibodies
Primary antibodies

Inhibitors & Agonists

est64454 hydrochloride

" in TargetMol Product Catalog

Inhibitors & Agonists
3

EST64454 hydrochloride

T88341950569-11-5

EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.

Sigma receptor

In Stock

Size

QTY

EST64454 free base

T709081351438-26-0

EST64454 is a σ1 receptor (σ1R) antagonist clinical candidate for the treatment of pain. EST64454 shows an outstanding aqueous solubility, which together with its high permeability in Caco-2 cells will allow its classification as a BCS class I compound. It also shows high metabolic stability.

Others

$1,520

1-2 weeks

Size

QTY

EST64454 Maleic acid salt

T93062088272-67-5

EST64454 Maleic acid salt is the maleic acid salt form of EST64454.EST64454 is a highly soluble σ1 receptor antagonist clinical candidate for the treatment of pain.

Others

In Stock

Size

QTY

Go to page 1

Page of 1

Catalog No.

Pack Size

Quantity

Name *

Organization *

Email *

Phone Number

Head of the research group/department

Official Quote Attachment *

Receiving country *

Remark

Product Comparison

Product
Species
Expression System
Tag
Accession Number
Amino Acid
Construction
Molecular Weight
Endotoxin
Formulation
Reconstitution
Stability & Storage
Shipping
Research Background
Size