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firazorexton

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Firazorexton
T398082274802-95-6
Firazorexton is a potent orexin type 2 receptor (OX2R) agonist.
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Firazorexton hydrate
TAK-994
T786362861934-86-1
Firazorexton hydrate (TAK-994) is a brain-penetrant, orally active agonist of the orexin type 2 receptor (OX2R) with a potent EC50 of 19 nM, effectively reducing wakefulness fragmentation and cataplexy-like episodes in mouse models of narcolepsy [1].
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8-10 weeks
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