T15943 |
M443
|
1820684-31-8
|
98%
|
|
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
|
T11286 |
Fiduxosin
|
208993-54-8
|
98%
|
|
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
|
T11010 |
Detomidine carboxylic acid
|
115664-39-6
|
98%
|
|
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
|
TN5061 |
Stephanine
|
517-63-5
|
98%
|
|
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
|
T1769 |
Pardoprunox
|
269718-84-5
|
98%
|
|
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
|
T14287 |
Ancarolol
|
75748-50-4
|
98%
|
|
Ancarolol is a blocking agent of beta-adrenergic.
|
T6860 |
ICI-118551 Hydrochloride
|
1217094-53-5
|
98%
|
|
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
|
T10778 |
CGP 20712 A
|
105737-62-0
|
98%
|
|
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
|
TN3507 |
Beta-Yohimbine
|
549-84-8
|
98%
|
|
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
|
T11036 |
Diacetolol D7
|
1346604-19-0
|
98%
|
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
|
T6562 |
Latrepirdine dihydrochloride
|
97657-92-6
|
98%
|
|
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
|
T11894 |
Lusaperidone
|
214548-46-6
|
98%
|
|
Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
|
T13285 |
Vatinoxan hydrochloride
|
130466-38-5
|
98%
|
|
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
|
T12815 |
(S)-Terazosin
|
109351-33-9
|
98%
|
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
|
T11786 |
KUL-7211 racemate
|
911196-40-2
|
98%
|
|
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
|
T10364 |
Arbutamine
|
128470-16-6
|
98%
|
|
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
T16769 |
Ro 363
|
74513-77-2
|
98%
|
|
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
|
T6663 |
Scopine hydrochloride
|
85700-55-6
|
98%
|
|
Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
|
T13403 |
ZK-90055 hydrochloride
|
84638-81-3
|
98%
|
|
ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
|