Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T15943	M443	1820684-31-8	98%
T15943	M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T11286	Fiduxosin	208993-54-8	98%
T11286	Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
T11010	Detomidine carboxylic acid	115664-39-6	98%
T11010	Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
TN5061	Stephanine	517-63-5	98%
TN5061	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T1769	Pardoprunox	269718-84-5	98%
T1769	Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T14287	Ancarolol	75748-50-4	98%
T14287	Ancarolol is a blocking agent of beta-adrenergic.
T6860	ICI-118551 Hydrochloride	1217094-53-5	98%
T6860	ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T10778	CGP 20712 A	105737-62-0	98%
T10778	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
TN3507	Beta-Yohimbine	549-84-8	98%
TN3507	Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T11036	Diacetolol D7	1346604-19-0	98%
T11036	Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T6562	Latrepirdine dihydrochloride	97657-92-6	98%
T6562	Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T11894	Lusaperidone	214548-46-6	98%
T11894	Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
T13285	Vatinoxan hydrochloride	130466-38-5	98%
T13285	Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T12815	(S)-Terazosin	109351-33-9	98%
T12815	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T11786	KUL-7211 racemate	911196-40-2	98%
T11786	KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
T10364	Arbutamine	128470-16-6	98%
T10364	Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
TN3368	Akuammigine	642-17-1	98%
TN3368	Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T16769	Ro 363	74513-77-2	98%
T16769	RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
T6663	Scopine hydrochloride	85700-55-6	98%
T6663	Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
T13403	ZK-90055 hydrochloride	84638-81-3	98%
T13403	ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.