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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T10066 2',5'-Dideoxyadenosine 6698-26-6 98.66%
2',5'-Dideoxyadenosine
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
T14490 Talipexole dihydrochloride 36085-73-1 98.64%
Talipexole dihydrochloride
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
T22612 BMY-14802 hydrochloride 105565-55-7 98.64%
BMY-14802 hydrochloride
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
T20157 Brimonidine 59803-98-4 98.60%
Brimonidine
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
T2535 Ivabradine hydrochloride 148849-67-6 98.6%
Ivabradine hydrochloride
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioav...
T22369 Midodrine 42794-76-3 98.57%
Midodrine
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
T13804 OPC-28326 167626-17-7 98.56%
OPC-28326
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
T31175 Dabelotine 118976-38-8 98.55%
Dabelotine
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
T8899 Metipranolol 22664-55-7 98.54%
Metipranolol
Metipranolol is a useful organic compound for research related to life sciences. The catalog number is T8899 and the CAS number is 22664-55-7.
T26923 Bunazosin Hydrochloride 52712-76-2 98.48%
Bunazosin Hydrochloride
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
T10952 Dabuzalgron 219311-44-1 98.47%
Dabuzalgron
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
T68124 Pafenolol 75949-61-0 98.43%
Pafenolol
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.
T7079 Batefenterol 743461-65-6 98.4%
Batefenterol
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
T17111 Todralazine hydrochloride 3778-76-5 98.32%
Todralazine hydrochloride
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can b...
T11095L DREADD agonist 21 56296-18-5 98.27%
DREADD agonist 21
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T6653 Salmeterol Xinafoate 94749-08-3 98.24%
Salmeterol Xinafoate
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma sympto...
T28895 T-0509 96843-99-1 98.21%
T-0509
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-adrenoceptor...
T33386 Milveterol HCl 804518-03-4 98.2%
Milveterol HCl
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
T68023L Tolnapersine TFA T68023L 98.10%
Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
T11148 Ecastolol 77695-52-4 98.1%
Ecastolol
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
2',5'-Dideoxyadenosine
T10066
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
Talipexole dihydrochloride
T14490
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
BMY-14802 hydrochloride
T22612
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
Brimonidine
T20157
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
Ivabradine hydrochloride
T2535
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioav...
Midodrine
T22369
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
OPC-28326
T13804
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
Dabelotine
T31175
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
Metipranolol
T8899
Metipranolol is a useful organic compound for research related to life sciences. The catalog number is T8899 and the CAS number is 22664-55-7.
Bunazosin Hydrochloride
T26923
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
Dabuzalgron
T10952
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
Pafenolol
T68124
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.
Batefenterol
T7079
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
Todralazine hydrochloride
T17111
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can b...
DREADD agonist 21
T11095L
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
Salmeterol Xinafoate
T6653
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma sympto...
T-0509
T28895
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-adrenoceptor...
Milveterol HCl
T33386
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
Tolnapersine TFA
T68023L
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Ecastolol
T11148
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
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TargetMol