Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T8149	Dobutamine hydrochloride	49745-95-1	98.52%
T8149	Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T26923	Bunazosin Hydrochloride	52712-76-2	98.48%
T26923	Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
T10952	Dabuzalgron	219311-44-1	98.47%
T10952	Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
T6562	Latrepirdine dihydrochloride	97657-92-6	98.45%
T6562	Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
T6519	Gramine	87-52-5	98.44%
T6519	Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
T68124	Pafenolol	75949-61-0	98.43%
T68124	Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.
T26778L	Besipirdine hydrochloride	130953-69-4	98.40%
T26778L	Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine hydrochloride inhib...
T7079	Batefenterol	743461-65-6	98.4%
T7079	Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
T17111	Todralazine hydrochloride	3778-76-5	98.32%
T17111	Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can b...
T11095L	DREADD agonist 21	56296-18-5	98.27%
T11095L	DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T6653	Salmeterol Xinafoate	94749-08-3	98.24%
T6653	Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma sympto...
T28895	T-0509	96843-99-1	98.21%
T28895	T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-adrenoceptor...
T33386	Milveterol HCl	804518-03-4	98.2%
T33386	Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
T10250	ADRA1D receptor antagonist 1 HCl	1191908-14-1	98.13%
T10250	ADRA1D receptor antagonist 1 HCl is an orally active, potent and selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activ...
T68023L	Tolnapersine TFA	T68023L	98.10%
T68023L	Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
T11148	Ecastolol	77695-52-4	98.1%
T11148	Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
TN7129	Methyl maslinate	22425-82-7	98.1%
TN7129	Methyl maslinate (Maslinic acid methyl ester) is an antagonist of β- adrenergic receptor with cardiotonic and antidysrhythmic properties. Methyl maslinate can be...
T0397	Tetrahydrozoline	84-22-0	98.07%
T0397	Tetrahydrozoline (Tetryzoline), an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of th...
TP1902L1	G-Protein antagonist peptide acetate	TP1902L1	98.06%
TP1902L1	G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide aceta...
T1158	Phenoxybenzamine hydrochloride	63-92-3	98.04%
T1158	Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...