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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
TN3507 Beta-Yohimbine 549-84-8 98%
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T10778 CGP 20712 A 105737-62-0 98%
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
T6860 ICI-118551 Hydrochloride 1217094-53-5 98%
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T14287 Ancarolol 75748-50-4 98%
Ancarolol is a blocking agent of beta-adrenergic.
TN5061 Stephanine 517-63-5 98%
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T11010 Detomidine carboxylic acid 115664-39-6 98%
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T68023 Tolnapersine 70312-00-4 98%
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
T11286 Fiduxosin 208993-54-8 98%
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
T15943 M443 1820684-31-8 98%
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T0101 Doxazosin mesylate 77883-43-3 99.98%
Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T1282 Carteolol hydrochloride 51781-21-6 99.97%
Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
T21066 Norepinephrine bitartrate salt 3414-63-9 99.97%
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T1539 Iloperidone 133454-47-4 99.96%
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T9220 Naftopidil hydrochloride 1164469-60-6 99.95%
Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocepto...
T5511 L-765314 189349-50-6 99.95%
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
T0210L Tamsulosin 106133-20-4 99.94%
Tansulosin is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulosin is used to treat difficul...
T0455 Clozapine 5786-21-0 99.93%
Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
T17310 Phenylephrine 59-42-7 99.92%
Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T0103 Dipivefrin hydrochloride 64019-93-8 99.92%
Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T1073 Dronedarone hydrochloride 141625-93-6 99.91%
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
beta-Yohimbine
TN3507
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
CGP 20712 A
T10778
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
ICI-118551 Hydrochloride
T6860
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
Ancarolol
T14287
Ancarolol is a blocking agent of beta-adrenergic.
Stephanine
TN5061
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
Detomidine carboxylic acid
T11010
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
Tolnapersine
T68023
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Fiduxosin
T11286
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
M443
T15943
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
Doxazosin mesylate
T0101
Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
Carteolol hydrochloride
T1282
Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
Norepinephrine bitartrate salt
T21066
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
Iloperidone
T1539
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Naftopidil hydrochloride
T9220
Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocepto...
L-765314
T5511
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
Tamsulosin
T0210L
Tansulosin is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulosin is used to treat difficul...
Clozapine
T0455
Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
Phenylephrine
T17310
Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
Dipivefrin hydrochloride
T0103
Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
Dronedarone hydrochloride
T1073
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
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