TN3507 |
Beta-Yohimbine
|
549-84-8
|
98%
|
|
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
|
T10778 |
CGP 20712 A
|
105737-62-0
|
98%
|
|
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
|
T6860 |
ICI-118551 Hydrochloride
|
1217094-53-5
|
98%
|
|
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
|
T14287 |
Ancarolol
|
75748-50-4
|
98%
|
|
Ancarolol is a blocking agent of beta-adrenergic.
|
TN5061 |
Stephanine
|
517-63-5
|
98%
|
|
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
|
T11010 |
Detomidine carboxylic acid
|
115664-39-6
|
98%
|
|
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
|
T68023 |
Tolnapersine
|
70312-00-4
|
98%
|
|
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
|
T11286 |
Fiduxosin
|
208993-54-8
|
98%
|
|
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
|
T15943 |
M443
|
1820684-31-8
|
98%
|
|
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
|
T0101 |
Doxazosin mesylate
|
77883-43-3
|
99.98%
|
|
Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
|
T1282 |
Carteolol hydrochloride
|
51781-21-6
|
99.97%
|
|
Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
|
T21066 |
Norepinephrine bitartrate salt
|
3414-63-9
|
99.97%
|
|
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
|
T1539 |
Iloperidone
|
133454-47-4
|
99.96%
|
|
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
|
T9220 |
Naftopidil hydrochloride
|
1164469-60-6
|
99.95%
|
|
Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocepto...
|
T5511 |
L-765314
|
189349-50-6
|
99.95%
|
|
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
|
T0210L |
Tamsulosin
|
106133-20-4
|
99.94%
|
|
Tansulosin is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulosin is used to treat difficul...
|
T0455 |
Clozapine
|
5786-21-0
|
99.93%
|
|
Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
|
T17310 |
Phenylephrine
|
59-42-7
|
99.92%
|
|
Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
|
T0103 |
Dipivefrin hydrochloride
|
64019-93-8
|
99.92%
|
|
Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
|
T1073 |
Dronedarone hydrochloride
|
141625-93-6
|
99.91%
|
|
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
|