Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
TN3507	Beta-Yohimbine	549-84-8	98%
TN3507	Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T10778	CGP 20712 A	105737-62-0	98%
T10778	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
T6860	ICI-118551 Hydrochloride	1217094-53-5	98%
T6860	ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T14287	Ancarolol	75748-50-4	98%
T14287	Ancarolol is a blocking agent of beta-adrenergic.
TN5061	Stephanine	517-63-5	98%
TN5061	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T11010	Detomidine carboxylic acid	115664-39-6	98%
T11010	Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T68023	Tolnapersine	70312-00-4	98%
T68023	Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
T11286	Fiduxosin	208993-54-8	98%
T11286	Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
T15943	M443	1820684-31-8	98%
T15943	M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T0101	Doxazosin mesylate	77883-43-3	99.98%
T0101	Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T1282	Carteolol hydrochloride	51781-21-6	99.97%
T1282	Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
T21066	Norepinephrine bitartrate salt	3414-63-9	99.97%
T21066	Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T1539	Iloperidone	133454-47-4	99.96%
T1539	Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T9220	Naftopidil hydrochloride	1164469-60-6	99.95%
T9220	Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocepto...
T5511	L-765314	189349-50-6	99.95%
T5511	L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
T0210L	Tamsulosin	106133-20-4	99.94%
T0210L	Tansulosin is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulosin is used to treat difficul...
T0455	Clozapine	5786-21-0	99.93%
T0455	Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
T17310	Phenylephrine	59-42-7	99.92%
T17310	Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T0103	Dipivefrin hydrochloride	64019-93-8	99.92%
T0103	Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T1073	Dronedarone hydrochloride	141625-93-6	99.91%
T1073	Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.