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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T20570 Labetalol 36894-69-6 99.87%
Labetalol
Labetalol (Apo-Labetalol) is a mixed alpha/beta-adrenergic antagonist.It is used to treat high blood pressure. It can be given by mouth for long term hypertensio...
T1050 Prazosin hydrochloride 19237-84-4 99.87%
Prazosin hydrochloride
Prazosin hydrochloride (Vasoflex) reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism n...
T0290 Tizanidine hydrochloride 64461-82-1 99.87%
Tizanidine hydrochloride
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
T8348 Phentolamine 50-60-2 99.86%
Phentolamine
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T0993 Methoxamine hydrochloride 61-16-5 99.86%
Methoxamine hydrochloride
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T0505 Methyldopa 555-30-6 99.86%
Methyldopa
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic...
T8738 LUN42518 HCl 47142-51-8(free base) T8738 99.85%
LUN42518 HCl  47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
T0469 Octopamine hydrochloride 770-05-8 99.85%
Octopamine hydrochloride
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a ne...
T3275 Nefazodone hydrochloride 82752-99-6 99.85%
Nefazodone hydrochloride
Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.
T40622 Mapenterol hydrochloride 54238-51-6 99.85%
Mapenterol hydrochloride
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
T22316 Doxazosin 74191-85-8 99.85%
Doxazosin
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
T0154 Nebivolol hydrochloride 152520-56-4 99.85%
Nebivolol hydrochloride
Nebivolol hydrochloride (R 065824 hydrochloride) is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR throug...
T30140 Arotinolol hydrochloride 68377-91-3 99.84%
Arotinolol hydrochloride
Arotinolol hydrochloride(Arotinolol HCl) is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I...
T0115 Idazoxan hydrochloride 79944-56-2 99.84%
Idazoxan hydrochloride
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T6422 Brimonidine Tartrate 70359-46-5 99.83%
Brimonidine Tartrate
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pres...
T0277 Metaproterenol hemisulfate 5874-97-5 99.83%
Metaproterenol hemisulfate
Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
T6522 Guanabenz Acetate 23256-50-0 99.83%
Guanabenz Acetate
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic rece...
T23557 Talibegron hydrochloride 178600-17-4 99.82%
Talibegron hydrochloride
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Re...
T5S2178 Fargesin 31008-19-2 99.82%
Fargesin
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Far...
T68129L1 Picumeterol FA 99.80%
Picumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist. In in vitro and in vivo tests, picumeterol FA produces long-lasting airway smooth muscle...
Labetalol
T20570
Labetalol (Apo-Labetalol) is a mixed alpha/beta-adrenergic antagonist.It is used to treat high blood pressure. It can be given by mouth for long term hypertensio...
Prazosin hydrochloride
T1050
Prazosin hydrochloride (Vasoflex) reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism n...
Tizanidine hydrochloride
T0290
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Phentolamine
T8348
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
Methoxamine hydrochloride
T0993
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
Methyldopa
T0505
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic...
LUN42518 HCl 47142-51-8(free base)
T8738
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
Octopamine hydrochloride
T0469
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a ne...
Nefazodone hydrochloride
T3275
Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.
Mapenterol hydrochloride
T40622
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
Doxazosin
T22316
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
Nebivolol hydrochloride
T0154
Nebivolol hydrochloride (R 065824 hydrochloride) is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR throug...
Arotinolol hydrochloride
T30140
Arotinolol hydrochloride(Arotinolol HCl) is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I...
Idazoxan hydrochloride
T0115
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
Brimonidine Tartrate
T6422
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pres...
Metaproterenol hemisulfate
T0277
Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
Guanabenz Acetate
T6522
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic rece...
Talibegron hydrochloride
T23557
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Re...
Fargesin
T5S2178
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Far...
Picumeterol FA
T68129L1
picumeterol FA is a potent and selective β2-adrenergic receptor agonist. In in vitro and in vivo tests, picumeterol FA produces long-lasting airway smooth muscle...
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TargetMol