Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T30140	Arotinolol hydrochloride	68377-91-3	99.84%
T30140	Arotinolol hydrochloride（Arotinolol HCl） is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I...
T7044	Norepinephrine	51-41-2	99.84%
T7044	Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression ...
T0115	Idazoxan hydrochloride	79944-56-2	99.84%
T0115	Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0042	Xylometazoline hydrochloride	1218-35-5	99.83%
T0042	Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.
T6422	Brimonidine Tartrate	70359-46-5	99.83%
T6422	Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pres...
T0277	Metaproterenol hemisulfate	5874-97-5	99.83%
T0277	Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
T23382	Spiroxatrine	1054-88-2	99.83%
T23382	Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2,...
T6522	Guanabenz Acetate	23256-50-0	99.83%
T6522	Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic rece...
T23557	Talibegron hydrochloride	178600-17-4	99.82%
T23557	Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Re...
T5S2178	Fargesin	31008-19-2	99.82%
T5S2178	1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Far...
T3033	Deoxycorticosterone acetate	56-47-3	99.81%
T3033	Deoxycorticosterone acetate (Cortexone acetate) is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of...
T23230	Rec 15/2615 dihydrochloride	173059-17-1	99.81%
T23230	Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.
T68129L1	Picumeterol FA		99.80%
T68129L1	picumeterol FA is a potent and selective β2-adrenergic receptor agonist. In in vitro and in vivo tests, picumeterol FA produces long-lasting airway smooth muscle...
T0852	Carbazochrome sodium sulfonate	51460-26-5	99.8%
T0852	Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
T1247	Clonidine hydrochloride	4205-91-8	99.8%
T1247	Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
T23536	Xamoterol hemifumarate	73210-73-8	99.79%
T23536	Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationship between...
T1186L	Ifenprodil	23210-56-2	99.78%
T1186L	Ifenprodil (RC61-91) is an inhibitor of the NMDA receptor, specifically of GluN1 (glycine-binding NMDA receptor subunit 1) and GluN2B (glutamate-binding NMDA rec...
T22245	Arformoterol Tartrate	200815-49-2	99.78%
T22245	Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol. Arformoterol is a long-acting beta-2 adrenergic agonist with bronchodilat...
T11318	Dopexamine hydrochloride	86484-91-5	99.77%
T11318	Dopexamine hydrochloride (FPL60278AR) is a β2-adrenergic receptor agonist. Dopexamine can attenuate the inflammatory response and protect against organ injury in...
T22029	AL 34662	210580-75-9	99.77%
T22029	AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a lo...