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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T21446 Rotigotine Hydrochloride 125572-93-2 99.53%
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T0031L2 Ziprasidone 146939-27-7 99.53%
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T3033 Deoxycorticosterone acetate 56-47-3 99.53%
Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
TN1922 Meranzin hydrate 5875-49-0 99.49%
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
T2889 Isoferulic acid 537-73-5 99.49%
3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
T22882 JP1302 80259-18-3 99.48%
JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.JP1302 has antidepressant activity, disrupts...
T13016 SR59230A 174689-39-5 99.46%
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T28267 ORM-10921 610782-82-6 99.46%
ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
T30586L Brefonalol HCl 99.45%
Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
T77565 Fluparoxan hydrochloride 105227-44-9 99.44%
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
T6408 Betaxolol 63659-18-7 99.43%
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T13376 YS-49 132836-42-1 99.42%
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T5S2059 Glaucine 475-81-0 99.42%
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T6652 Salbutamol hemisulfate 51022-70-9 99.39%
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T4983 Isoetharine mesylate salt 7279-75-6 99.35%
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T10830 CL 316243 138908-40-4 99.34%
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
T1239 Indacaterol maleate 753498-25-8 99.31%
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T0137 Mirtazapine 85650-52-8 99.3%
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T16798 RS 17053 hydrochloride 169505-93-5 99.27%
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T9762 Upidosin 152735-23-4 99.26%
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
Rotigotine Hydrochloride
T21446
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
Ziprasidone
T0031L2
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Deoxycorticosterone acetate
T3033
Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
Meranzin hydrate
TN1922
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
Isoferulic acid
T2889
3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
JP1302
T22882
JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.JP1302 has antidepressant activity, disrupts...
SR59230A
T13016
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
ORM-10921
T28267
ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
Brefonalol HCl
T30586L
Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
Fluparoxan hydrochloride
T77565
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
Betaxolol
T6408
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
YS-49
T13376
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
Glaucine
T5S2059
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
Salbutamol hemisulfate
T6652
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
Isoetharine mesylate salt
T4983
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
CL 316243
T10830
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
Indacaterol maleate
T1239
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
RS 17053 hydrochloride
T16798
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
Upidosin
T9762
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
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