Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T21446	Rotigotine Hydrochloride	125572-93-2	99.53%
T21446	Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T0031L2	Ziprasidone	146939-27-7	99.53%
T0031L2	Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T3033	Deoxycorticosterone acetate	56-47-3	99.53%
T3033	Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
TN1922	Meranzin hydrate	5875-49-0	99.49%
TN1922	Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
T2889	Isoferulic acid	537-73-5	99.49%
T2889	3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
T22882	JP1302	80259-18-3	99.48%
T22882	JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.JP1302 has antidepressant activity, disrupts...
T13016	SR59230A	174689-39-5	99.46%
T13016	SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T28267	ORM-10921	610782-82-6	99.46%
T28267	ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
T30586L	Brefonalol HCl		99.45%
T30586L	Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
T77565	Fluparoxan hydrochloride	105227-44-9	99.44%
T77565	Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
T6408	Betaxolol	63659-18-7	99.43%
T6408	Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T13376	YS-49	132836-42-1	99.42%
T13376	YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T5S2059	Glaucine	475-81-0	99.42%
T5S2059	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T6652	Salbutamol hemisulfate	51022-70-9	99.39%
T6652	Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T4983	Isoetharine mesylate salt	7279-75-6	99.35%
T4983	Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T10830	CL 316243	138908-40-4	99.34%
T10830	CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
T1239	Indacaterol maleate	753498-25-8	99.31%
T1239	Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T0137	Mirtazapine	85650-52-8	99.3%
T0137	Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T16798	RS 17053 hydrochloride	169505-93-5	99.27%
T16798	RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T9762	Upidosin	152735-23-4	99.26%
T9762	Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...