Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T10066	2',5'-Dideoxyadenosine	6698-26-6	98%
T10066	2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 µM).
T77566	(3aR,9aR)-Fluparoxan	105182-47-6	98%
T77566	(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
T8304	Anisodamine Hydrobromide	55449-49-5	98%
T8304	Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T3232	Higenamine hydrochloride	11041-94-4	98%
T3232	Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupl...
T13655	DL-Norepinephrine hydrochloride	55-27-6	98%
T13655	DL-Norepinephrine hydrochloride is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
T1696	2-(1-Piperazinyl)pyrimidine	20980-22-7	98%
T1696	2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
T24588	Palatrigine	98410-36-7	98%
T24588	Palatrigine is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.
T1738	Taxifolin	480-18-2	98%
T1738	Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
T30027	Amosulalol	85320-68-9	98%
T30027	Amosulalol is a combined alpha and beta adrenoceptor antagonist.
T12643	(R)-Terazosin	109351-34-0	98%
T12643	(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6....
T12970	Solabegron	252920-94-8	98%
T12970	Solabegron is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM...
T6653	Salmeterol Xinafoate	94749-08-3	98%
T6653	Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstruc...
T1139	Salbutamol	18559-94-9	98%
T1139	Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', ...
T2535	Ivabradine hydrochloride	148849-67-6	98%
T2535	Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyp...
T0270	Hydrocortisone 17-butyrate	13609-67-1	98%
T0270	Hydrocortisone Butyrate is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
T20898	(R)-Propranolol hydrochloride	13071-11-9	98%
T20898	(R)-(+)-PROPRANOLOL is a less active enantiomer of propranolol.
T8389	Trifluoperazine	117-89-5	98%
T8389	Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
T0453	Phenylephrine hydrochloride	61-76-7	98%
T0453	Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
T3046	BMY 7378 dihydrochloride	21102-95-4	98%
T3046	BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T7160	Lofexidine	31036-80-3	98%
T7160	Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.