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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T10066 2',5'-Dideoxyadenosine 6698-26-6 98%
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 µM).
T77566 (3aR,9aR)-Fluparoxan 105182-47-6 98%
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
T8304 Anisodamine Hydrobromide 55449-49-5 98%
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T3232 Higenamine hydrochloride 11041-94-4 98%
Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupl...
T13655 DL-Norepinephrine hydrochloride 55-27-6 98%
DL-Norepinephrine hydrochloride is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
T1696 2-(1-Piperazinyl)pyrimidine 20980-22-7 98%
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
T24588 Palatrigine 98410-36-7 98%
Palatrigine is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.
T1738 Taxifolin 480-18-2 98%
Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
T30027 Amosulalol 85320-68-9 98%
Amosulalol is a combined alpha and beta adrenoceptor antagonist.
T12643 (R)-Terazosin 109351-34-0 98%
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6....
T12970 Solabegron 252920-94-8 98%
Solabegron is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM...
T6653 Salmeterol Xinafoate 94749-08-3 98%
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstruc...
T1139 Salbutamol 18559-94-9 98%
Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', ...
T2535 Ivabradine hydrochloride 148849-67-6 98%
Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyp...
T0270 Hydrocortisone 17-butyrate 13609-67-1 98%
Hydrocortisone Butyrate is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
T20898 (R)-Propranolol hydrochloride 13071-11-9 98%
(R)-(+)-PROPRANOLOL is a less active enantiomer of propranolol.
T8389 Trifluoperazine 117-89-5 98%
Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
T0453 Phenylephrine hydrochloride 61-76-7 98%
Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
T3046 BMY 7378 dihydrochloride 21102-95-4 98%
BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T7160 Lofexidine 31036-80-3 98%
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
2',5'-Dideoxyadenosine
T10066
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 µM).
(3aR,9aR)-Fluparoxan
T77566
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
Anisodamine Hydrobromide
T8304
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Higenamine hydrochloride
T3232
Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupl...
DL-Norepinephrine hydrochloride
T13655
DL-Norepinephrine hydrochloride is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
2-(1-Piperazinyl)pyrimidine
T1696
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Palatrigine
T24588
Palatrigine is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.
Taxifolin
T1738
Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
Amosulalol
T30027
Amosulalol is a combined alpha and beta adrenoceptor antagonist.
(R)-Terazosin
T12643
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6....
Solabegron
T12970
Solabegron is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM...
Salmeterol Xinafoate
T6653
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstruc...
Salbutamol
T1139
Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', ...
Ivabradine hydrochloride
T2535
Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyp...
Hydrocortisone 17-butyrate
T0270
Hydrocortisone Butyrate is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
(R)-Propranolol hydrochloride
T20898
(R)-(+)-PROPRANOLOL is a less active enantiomer of propranolol.
Trifluoperazine
T8389
Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
Phenylephrine hydrochloride
T0453
Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
BMY 7378 dihydrochloride
T3046
BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
Lofexidine
T7160
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
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