Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T3284	Carazolol	57775-29-8	98%
T3284	Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T2226	Pergolide mesylate	66104-23-2	98%
T2226	PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
T0445	Promethazine	60-87-7	98%
T0445	Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
T7046	Xylazine	7361-61-7	98%
T7046	Xylazine is α2-adrenergic receptor agonist.
T3431	Pardoprunox hydrochloride	269718-83-4	98%
T3431	Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6...
T23283	2-Methoxyidazoxan monohydrochloride	109544-45-8	98%
T23283	α2-adrenoceptor antagonist
T1671	Mirabegron	223673-61-8	98%
T1671	Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T21640	Talinolol	57460-41-0	98%
T21640	(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T21445	Naphazoline	835-31-4	98%
T21445	Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
T9762	Upidosin	152735-23-4	98%
T9762	Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
T16798	RS 17053 hydrochloride	169505-93-5	98%
T16798	RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T22406	Prazosin	19216-56-9	98%
T22406	Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T0348	Labetalol hydrochloride	32780-64-6	98%
T0348	Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
T0324	Isoxsuprine hydrochloride	579-56-6	98%
T0324	Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0137	Mirtazapine	85650-52-8	98%
T0137	Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T0031L	Ziprasidone hydrochloride	122883-93-6	98%
T0031L	Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T4983	Isoetharine mesylate salt	7279-75-6	98%
T4983	Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T1577	Midodrine hydrochloride	3092-17-9	98%
T1577	Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
T6652	Salbutamol hemisulfate	51022-70-9	98%
T6652	Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T0696	Naftopidil	57149-07-2	98%
T0696	Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.