T3284 |
Carazolol
|
57775-29-8
|
98%
|
|
Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
|
T2226 |
Pergolide mesylate
|
66104-23-2
|
98%
|
|
PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
|
T0445 |
Promethazine
|
60-87-7
|
98%
|
|
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
|
T7046 |
Xylazine
|
7361-61-7
|
98%
|
|
Xylazine is α2-adrenergic receptor agonist.
|
T3431 |
Pardoprunox hydrochloride
|
269718-83-4
|
98%
|
|
Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6...
|
T23283 |
2-Methoxyidazoxan monohydrochloride
|
109544-45-8
|
98%
|
|
α2-adrenoceptor antagonist
|
T1671 |
Mirabegron
|
223673-61-8
|
98%
|
|
Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
|
T21640 |
Talinolol
|
57460-41-0
|
98%
|
|
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
|
T21445 |
Naphazoline
|
835-31-4
|
98%
|
|
Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
|
T9762 |
Upidosin
|
152735-23-4
|
98%
|
|
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
|
T16798 |
RS 17053 hydrochloride
|
169505-93-5
|
98%
|
|
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
|
T22406 |
Prazosin
|
19216-56-9
|
98%
|
|
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
|
T0348 |
Labetalol hydrochloride
|
32780-64-6
|
98%
|
|
Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
|
T0324 |
Isoxsuprine hydrochloride
|
579-56-6
|
98%
|
|
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
|
T0137 |
Mirtazapine
|
85650-52-8
|
98%
|
|
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
|
T0031L |
Ziprasidone hydrochloride
|
122883-93-6
|
98%
|
|
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
|
T4983 |
Isoetharine mesylate salt
|
7279-75-6
|
98%
|
|
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
|
T1577 |
Midodrine hydrochloride
|
3092-17-9
|
98%
|
|
Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
|
T6652 |
Salbutamol hemisulfate
|
51022-70-9
|
98%
|
|
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
|
T0696 |
Naftopidil
|
57149-07-2
|
98%
|
|
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
|