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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T3284 Carazolol 57775-29-8 98%
Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T2226 Pergolide mesylate 66104-23-2 98%
PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
T0445 Promethazine 60-87-7 98%
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
T7046 Xylazine 7361-61-7 98%
Xylazine is α2-adrenergic receptor agonist.
T3431 Pardoprunox hydrochloride 269718-83-4 98%
Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6...
T23283 2-Methoxyidazoxan monohydrochloride 109544-45-8 98%
α2-adrenoceptor antagonist
T1671 Mirabegron 223673-61-8 98%
Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T21640 Talinolol 57460-41-0 98%
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T21445 Naphazoline 835-31-4 98%
Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
T9762 Upidosin 152735-23-4 98%
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
T16798 RS 17053 hydrochloride 169505-93-5 98%
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T22406 Prazosin 19216-56-9 98%
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T0348 Labetalol hydrochloride 32780-64-6 98%
Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
T0324 Isoxsuprine hydrochloride 579-56-6 98%
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0137 Mirtazapine 85650-52-8 98%
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T0031L Ziprasidone hydrochloride 122883-93-6 98%
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T4983 Isoetharine mesylate salt 7279-75-6 98%
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T1577 Midodrine hydrochloride 3092-17-9 98%
Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
T6652 Salbutamol hemisulfate 51022-70-9 98%
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T0696 Naftopidil 57149-07-2 98%
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
Carazolol
T3284
Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
Pergolide mesylate
T2226
PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
Promethazine
T0445
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
Xylazine
T7046
Xylazine is α2-adrenergic receptor agonist.
Pardoprunox hydrochloride
T3431
Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6...
2-Methoxyidazoxan monohydrochloride
T23283
α2-adrenoceptor antagonist
Mirabegron
T1671
Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
Talinolol
T21640
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Naphazoline
T21445
Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
Upidosin
T9762
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM...
RS 17053 hydrochloride
T16798
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
Prazosin
T22406
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Labetalol hydrochloride
T0348
Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
Isoxsuprine hydrochloride
T0324
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Ziprasidone hydrochloride
T0031L
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Isoetharine mesylate salt
T4983
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
Midodrine hydrochloride
T1577
Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
Salbutamol hemisulfate
T6652
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
Naftopidil
T0696
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
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