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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T5S2059 Glaucine 475-81-0 98%
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T13376 YS-49 132836-42-1 98%
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T77565 Fluparoxan hydrochloride 105227-44-9 98%
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
T10998 Deriglidole 122830-14-2 98%
Deriglidole is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does...
T30586L Brefonalol HCl 98%
Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
T2645 Vilanterol 503068-34-6 98%
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
T13016 SR59230A 174689-39-5 98%
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T1503 Esmolol hydrochloride 81161-17-3 98%
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
T2889 Isoferulic acid 537-73-5 98%
3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
TN1922 Meranzin hydrate 5875-49-0 98%
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
T1056 Isoprenaline hydrochloride 51-30-9 98%
Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
T0351 Risperidone 106266-06-2 98%
Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T6408 Betaxolol 63659-18-7 98%
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T0031L2 Ziprasidone 146939-27-7 98%
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T0279 Metaraminol tartrate 33402-03-8 98%
Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the...
T11607 ICI 118,551 hydrochloride 72795-01-8 98%
ICI 118,551 is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3 receptors).
T0365 Thioridazine hydrochloride 130-61-0 98%
Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
T7056 Dronedarone 141626-36-0 98%
Dronedarone is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T0226 Betaxolol hydrochloride 63659-19-8 98%
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
T6241 Quetiapine hemifumarate 111974-72-2 98%
Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
Glaucine
T5S2059
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
YS-49
T13376
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
Fluparoxan hydrochloride
T77565
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
Deriglidole
T10998
Deriglidole is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does...
Brefonalol HCl
T30586L
Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
Vilanterol
T2645
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
SR59230A
T13016
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
Esmolol hydrochloride
T1503
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
Isoferulic acid
T2889
3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
Meranzin hydrate
TN1922
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
Isoprenaline hydrochloride
T1056
Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
Risperidone
T0351
Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
Betaxolol
T6408
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
Ziprasidone
T0031L2
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Metaraminol tartrate
T0279
Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the...
ICI 118,551 hydrochloride
T11607
ICI 118,551 is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3 receptors).
Thioridazine hydrochloride
T0365
Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
Dronedarone
T7056
Dronedarone is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
Betaxolol hydrochloride
T0226
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
Quetiapine hemifumarate
T6241
Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
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