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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T0031L Ziprasidone hydrochloride 122883-93-6 99.34%
Ziprasidone hydrochloride
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
T10830 CL 316243 138908-40-4 99.34%
CL 316243
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
T1239 Indacaterol maleate 753498-25-8 99.31%
Indacaterol maleate
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
T0324 Isoxsuprine hydrochloride 579-56-6 99.31%
Isoxsuprine hydrochloride
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0137 Mirtazapine 85650-52-8 99.3%
Mirtazapine
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T22406 Prazosin 19216-56-9 99.29%
Prazosin
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T16798 RS 17053 hydrochloride 169505-93-5 99.27%
RS 17053 hydrochloride
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T9762 Upidosin 152735-23-4 99.26%
Upidosin
Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenocepto...
T21445 Naphazoline 835-31-4 99.25%
Naphazoline
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in ...
T6963 Reboxetine mesylate 98769-84-7 99.24%
Reboxetine mesylate
Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).
T10100 QF0301B 149247-12-1 99.16%
QF0301B
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
T21640 Talinolol 57460-41-0 99.15%
Talinolol
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T1671 Mirabegron 223673-61-8 99.14%
Mirabegron
Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T23283 2-Methoxyidazoxan monohydrochloride 109544-45-8 99.13%
2-Methoxyidazoxan monohydrochloride
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic eff...
T10631L Bucindolol Formate 99.11%
Bucindolol Formate
Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
T31750 Faxeladol 433265-65-7 99.11%
Faxeladol
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
T0445 Promethazine 60-87-7 99.11%
Promethazine
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
T2226 Pergolide mesylate 66104-23-2 99.09%
Pergolide mesylate
Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some...
T6872 L755507 159182-43-1 99.04%
L755507
L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
T8389 Trifluoperazine 117-89-5 99.03%
Trifluoperazine
Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
Ziprasidone hydrochloride
T0031L
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
CL 316243
T10830
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
Indacaterol maleate
T1239
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
Isoxsuprine hydrochloride
T0324
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
Mirtazapine
T0137
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
Prazosin
T22406
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
RS 17053 hydrochloride
T16798
RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
Upidosin
T9762
Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenocepto...
Naphazoline
T21445
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in ...
Reboxetine mesylate
T6963
Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).
QF0301B
T10100
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
Talinolol
T21640
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Mirabegron
T1671
Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
2-Methoxyidazoxan monohydrochloride
T23283
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic eff...
Bucindolol Formate
T10631L
Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
Faxeladol
T31750
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
Promethazine
T0445
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
Pergolide mesylate
T2226
Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some...
L755507
T6872
L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
Trifluoperazine
T8389
Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
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TargetMol