Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T5S2059	Glaucine	475-81-0	98%
T5S2059	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T13376	YS-49	132836-42-1	98%
T13376	YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T77565	Fluparoxan hydrochloride	105227-44-9	98%
T77565	Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
T10998	Deriglidole	122830-14-2	98%
T10998	Deriglidole is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does...
T30586L	Brefonalol HCl		98%
T30586L	Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
T2645	Vilanterol	503068-34-6	98%
T2645	Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
T13016	SR59230A	174689-39-5	98%
T13016	SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T1503	Esmolol hydrochloride	81161-17-3	98%
T1503	Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
T2889	Isoferulic acid	537-73-5	98%
T2889	3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
TN1922	Meranzin hydrate	5875-49-0	98%
TN1922	Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
T1056	Isoprenaline hydrochloride	51-30-9	98%
T1056	Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
T0351	Risperidone	106266-06-2	98%
T0351	Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T6408	Betaxolol	63659-18-7	98%
T6408	Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T0031L2	Ziprasidone	146939-27-7	98%
T0031L2	Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T0279	Metaraminol tartrate	33402-03-8	98%
T0279	Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the...
T11607	ICI 118,551 hydrochloride	72795-01-8	98%
T11607	ICI 118,551 is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3 receptors).
T0365	Thioridazine hydrochloride	130-61-0	98%
T0365	Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
T7056	Dronedarone	141626-36-0	98%
T7056	Dronedarone is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T0226	Betaxolol hydrochloride	63659-19-8	98%
T0226	Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
T6241	Quetiapine hemifumarate	111974-72-2	98%
T6241	Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.