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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T1459 Cisatracurium besylate 96946-42-8 98%
Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T5159 Olodaterol hydrochloride 869477-96-3 98%
Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and act...
T21957 Guanabenz hydrochloride 23113-43-1 98%
Guanabenz hydrochloride is an orally active α2-adrenoceptor agonist with hypotensive effects.
T4526 Piperoxan hydrochloride 135-87-5 98%
Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
T0091 Alfuzosin hydrochloride 81403-68-1 98%
Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
T10631L Bucindolol Formate 98%
Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
T34308 Rezatomidine 847829-38-3 98%
Rezatomidine is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.
T1632 Amitraz 33089-61-1 98%
AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic mang...
T22852 ICI 89406 53671-71-9 98%
β-adrenergic antagonist
T6688 Synephrine hydrochloride 5985-28-4 98%
SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T1239 Indacaterol maleate 753498-25-8 98%
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T1090 Perphenazine 58-39-9 98%
Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0783 Mianserin hydrochloride 21535-47-7 98%
Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
T1132 Nicergoline 27848-84-6 98%
Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T23397 ST 91 4749-61-5 98%
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
T2547 Droxidopa 23651-95-8 98%
Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auton...
T10168 5-HT1A modulator 1 142477-34-7 98%
5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
T10758L Centanafadine hydrochloride 923981-14-0 98%
Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83...
T21446 Rotigotine Hydrochloride 125572-93-2 98%
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T19680 Zotepine 26615-21-4 98%
Zotepine is a second-generation antipsychotic with a primary use as a treatment for schizophrenia, although clinical trials have been conducted into its efficacy...
Cisatracurium besylate
T1459
Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Olodaterol hydrochloride
T5159
Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and act...
Guanabenz hydrochloride
T21957
Guanabenz hydrochloride is an orally active α2-adrenoceptor agonist with hypotensive effects.
Piperoxan hydrochloride
T4526
Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
Alfuzosin hydrochloride
T0091
Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
Bucindolol Formate
T10631L
Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
Rezatomidine
T34308
Rezatomidine is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.
Amitraz
T1632
AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic mang...
ICI 89406
T22852
β-adrenergic antagonist
Synephrine hydrochloride
T6688
SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
Indacaterol maleate
T1239
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
Perphenazine
T1090
Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Mianserin hydrochloride
T0783
Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
Nicergoline
T1132
Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
ST 91
T23397
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
Droxidopa
T2547
Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auton...
5-HT1A modulator 1
T10168
5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
Centanafadine hydrochloride
T10758L
Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83...
Rotigotine Hydrochloride
T21446
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
Zotepine
T19680
Zotepine is a second-generation antipsychotic with a primary use as a treatment for schizophrenia, although clinical trials have been conducted into its efficacy...
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