Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T1459	Cisatracurium besylate	96946-42-8	98%
T1459	Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T5159	Olodaterol hydrochloride	869477-96-3	98%
T5159	Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and act...
T21957	Guanabenz hydrochloride	23113-43-1	98%
T21957	Guanabenz hydrochloride is an orally active α2-adrenoceptor agonist with hypotensive effects.
T4526	Piperoxan hydrochloride	135-87-5	98%
T4526	Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
T0091	Alfuzosin hydrochloride	81403-68-1	98%
T0091	Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
T10631L	Bucindolol Formate		98%
T10631L	Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
T34308	Rezatomidine	847829-38-3	98%
T34308	Rezatomidine is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.
T1632	Amitraz	33089-61-1	98%
T1632	AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic mang...
T22852	ICI 89406	53671-71-9	98%
T22852	β-adrenergic antagonist
T6688	Synephrine hydrochloride	5985-28-4	98%
T6688	SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T1239	Indacaterol maleate	753498-25-8	98%
T1239	Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T1090	Perphenazine	58-39-9	98%
T1090	Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0783	Mianserin hydrochloride	21535-47-7	98%
T0783	Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
T1132	Nicergoline	27848-84-6	98%
T1132	Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T23397	ST 91	4749-61-5	98%
T23397	ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
T2547	Droxidopa	23651-95-8	98%
T2547	Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auton...
T10168	5-HT1A modulator 1	142477-34-7	98%
T10168	5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
T10758L	Centanafadine hydrochloride	923981-14-0	98%
T10758L	Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83...
T21446	Rotigotine Hydrochloride	125572-93-2	98%
T21446	Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T19680	Zotepine	26615-21-4	98%
T19680	Zotepine is a second-generation antipsychotic with a primary use as a treatment for schizophrenia, although clinical trials have been conducted into its efficacy...