GluR

Glutamate receptors are synaptic and non synaptic receptors located primarily on the membranes of neuronal and glial cells.Glutamate receptors are responsible for the glutamate-mediated postsynaptic excitation of neural cells, and are important for neural communication, memory formation, learning, and regulation.

Cat. No.	Product name	CAS No.	Purity
T77581	KM02894	116850-74-9	98.72%
T77581	KM02894 is a glutamate release inhibitor. Cancer cells release high levels of glutamate that can disrupt normal bone turnover, which can lead to cancer-induced b...
T27949	LY382884	211566-75-5	98.71%
T27949	LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.
T16524	Philanthotoxin 74 dihydrochloride	1227301-51-0	98.6%
T16524	Philanthotoxin 74 dihydrochloride is an antagonist of AMPAR with IC50s of 263 and 296 nM for GluR3 and GluR1.
T9021	Ro0711401	714971-87-6	98.54%
T9021	Ro0711401 is an agonist of mGlu1 receptor.
T8434	SIB-1757	31993-01-8	98.49%
T8434	SIB-1757 (6-methyl-2-[(E)-phenyldiazenyl]pyridin-3) is a selective antagonist of mGlu5 metabotropic glutamate receptor subtype (hmGlu5, IC50 : 0.4 μM)
T6562	Latrepirdine dihydrochloride	97657-92-6	98.45%
T6562	Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
T9133	Caroverine hydrochloride	55750-05-5	98.37%
T9133	Caroverine hydrochloride (Caroverine HCL) is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. It is also an antioxidant and c...
T25853	NBQX Disodium	479347-86-9	98.22%
T25853	NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity. NBQX Disodium is a ...
T10809L	CHPG hydrochloride	T10809L	98.1%
T10809L	CHPG hydrochloride is a selective agonist of mGluR5.
T15456	GYKI 53655 hydrochloride	143692-48-2	98.02%
T15456	GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the study of neurological disorders.
T27828	Licostinel	153504-81-5	98.02%
T27828	Licostinel (CGP 63446) is a glutamate receptor antagonist. Licostinel protects against permanent focal cerebral ischemia.
T7292	FITM	932737-65-0	98%
T7292	FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).
T0256	Citric acid trilithium salt tetrahydrate	6080-58-6	98%
T0256	Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) , the active component of Lithium, is a medicine used in the therapy of psychiat...
T7579	1-BCP	34023-62-6	98%
T7579	1-BCP (Piperonylic acid piperidide) is a centrally active drug that modulates AMPA receptor gated currents.
T7178	CNQX	115066-14-3	98%
T7178	CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)
T0675	Topiramate	97240-79-4	98%
T0675	Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associate...
T7515	MTEP hydrochloride	1186195-60-7	98%
T7515	MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)
T5884	Chelidamic acid	138-60-3	98%
T5884	Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.
T3539	Lu AF21934	1445605-23-1	97.96%
T3539	Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).
T3010	Xanthurenic Acid	59-00-7	97.96%
T3010	Xanthurenic Acid (8-Hydroxykynurenic acid), a molecule arising from tryptophan metabolism by transamination of 3-hydroxykynurenine, activates mGlu2/3 Metabotropi...