Home Tools
Log in
Cart

Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T16476 PF-03654746 935840-31-6 99.1%
PF-03654746
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
TN3699 Corchoionoside C 185414-25-9 98%
Corchoionoside C
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T10770 Cetirizine D8 774596-22-4 98%
Cetirizine D8
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T77715 H4R antagonist 3 1003091-20-0 98%
H4R antagonist 3
H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of autoi...
T78126 Dothiepin 113-53-1 98%
Dothiepin
Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing nora...
T79786 H4R antagonist 2 1148115-99-4 98%
H4R antagonist 2
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid arthri...
T80645 4-Methylhistamine 36507-31-0 98%
4-Methylhistamine
4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and ...
T11729 JTE-952 1255303-54-8 98%
JTE-952
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
T15590 Iodophenpropit dihydrobromide 145196-87-8 98%
Iodophenpropit dihydrobromide
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
TN3483 Bakkenolide D 18456-03-6 98%
Bakkenolide D
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T12630 (R)-(-)-α-Methylhistamine dihydrobromide 868698-49-1 98%
(R)-(-)-α-Methylhistamine dihydrobromide
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN2155 Rhodiocyanoside A 168433-86-1 98%
Rhodiocyanoside A
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T11088 Doxepin D3 Hydrochloride 347840-07-7 98%
Doxepin D3 Hydrochloride
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
T15722 Lavoltidine 76956-02-0 98%
Lavoltidine
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T17118 Toreforant 952494-46-1 98%
Toreforant
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T12416 PF-03654746 Tosylate 1039399-17-1 98%
PF-03654746 Tosylate
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T12703 ReN-1869 hydrochloride 170149-76-5 98%
ReN-1869 hydrochloride
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T19443L N-Acetylhistamine acetate 98%
N-Acetylhistamine acetate
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
T2S0118 Daurinoline 2831-75-6 98%
Daurinoline
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12228 Niperotidine 84845-75-0 98%
Niperotidine
Niperotidine is an antagonist of histamine H2-receptor.
PF-03654746
T16476
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
Corchoionoside C
TN3699
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
Cetirizine D8
T10770
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
H4R antagonist 3
T77715
H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of autoi...
Dothiepin
T78126
Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing nora...
H4R antagonist 2
T79786
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid arthri...
4-Methylhistamine
T80645
4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and ...
JTE-952
T11729
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
Iodophenpropit dihydrobromide
T15590
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
Bakkenolide D
TN3483
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
(R)-(-)-α-Methylhistamine dihydrobromide
T12630
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
Rhodiocyanoside A
TN2155
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
Doxepin D3 Hydrochloride
T11088
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
Lavoltidine
T15722
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
Toreforant
T17118
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
PF-03654746 Tosylate
T12416
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
ReN-1869 hydrochloride
T12703
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
N-Acetylhistamine acetate
T19443L
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
Daurinoline
T2S0118
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
Niperotidine
T12228
Niperotidine is an antagonist of histamine H2-receptor.
1 2 3 4 5 6 7 8 9 10 11 12
TargetMol