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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T1336 Benztropine mesylate 132-17-2 100%
Benztropine mesylate
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISE...
T0903 Cinnarizine 298-57-7 100%
Cinnarizine
Cinnarizine (Stugeron) is a piperazine derivative having histamine H1-receptor and calcium-channel blocking activity with vasodilating and antiemetic properties ...
T0174 Cyproheptadine hydrochloride sesquihydrate 41354-29-4 100%
Cyproheptadine hydrochloride sesquihydrate
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
T1115 Doxylamine succinate 562-10-7 100%
Doxylamine succinate
Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties. Doxylamine succinate (Decapryn) competitively blocks the...
T2520 Desloratadine 100643-71-8 100%
Desloratadine
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typic...
T1269 Tripelennamine hydrochloride 154-69-8 100%
Tripelennamine hydrochloride
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
T0089 Cetirizine dihydrochloride 83881-52-1 100%
Cetirizine dihydrochloride
Cetirizine dihydrochloride (UCB P071) is an effective second-generation histamine H1 antagonist that is potent in the therapy of allergic rhinitis, confirmed urt...
T68146 Sufotidine 80343-63-1 100%
Sufotidine
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
T25875 Noberastine 110588-56-2 100%
Noberastine
Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.
T8599 Betazole dihydrochloride 138-92-1
Betazole dihydrochloride
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
T0994 Ketotifen fumarate 34580-14-8
Ketotifen fumarate
Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.
T5829 H4 Receptor antagonist 1 848217-00-5
H4 Receptor antagonist 1
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
T1278 Astemizole 68844-77-9
Astemizole
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 ...
T68122 Oxmetidine 72830-39-8 98%
Oxmetidine
Oxmetidine (SKF 92994) is a novel H2 receptor antagonist that is cytotoxic. Oxmetidine inhibits transmembrane calcium flux in cardiac and vascular tissues and is...
T0468 Lidocaine 137-58-6 98%
Lidocaine
Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation o...
T29096L Vapitadine 793655-64-8 98%
Vapitadine
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
T0383 Fenspiride hydrochloride 5053-08-7 98%
Fenspiride hydrochloride
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
TN1661 Ganoderic acid C2 103773-62-2 98%
Ganoderic acid C2
Ganoderic acid C2 has anti-inflammatory,and anti-tumor-promoting activities. Ganoderic acid C2 can inhibit histamine release, it also has inhibitory effects on t...
T20597 Alginic acid 9005-32-7 98%
Alginic acid
Alginic acid (Snow acid algin G) is a natural polysaccharide extracted from brown seaweeds with anti-anaphylactic and anti-inflammatory activities. Alginic acid ...
T4507 Chlorphenesin 104-29-0 98%
Chlorphenesin
Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.
Benztropine mesylate
T1336
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISE...
Cinnarizine
T0903
Cinnarizine (Stugeron) is a piperazine derivative having histamine H1-receptor and calcium-channel blocking activity with vasodilating and antiemetic properties ...
Cyproheptadine hydrochloride sesquihydrate
T0174
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
Doxylamine succinate
T1115
Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties. Doxylamine succinate (Decapryn) competitively blocks the...
Desloratadine
T2520
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typic...
Tripelennamine hydrochloride
T1269
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
Cetirizine dihydrochloride
T0089
Cetirizine dihydrochloride (UCB P071) is an effective second-generation histamine H1 antagonist that is potent in the therapy of allergic rhinitis, confirmed urt...
Sufotidine
T68146
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
Noberastine
T25875
Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.
Betazole dihydrochloride
T8599
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
Ketotifen fumarate
T0994
Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.
H4 Receptor antagonist 1
T5829
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
Astemizole
T1278
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 ...
Oxmetidine
T68122
Oxmetidine (SKF 92994) is a novel H2 receptor antagonist that is cytotoxic. Oxmetidine inhibits transmembrane calcium flux in cardiac and vascular tissues and is...
Lidocaine
T0468
Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation o...
Vapitadine
T29096L
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
Fenspiride hydrochloride
T0383
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
Ganoderic acid C2
TN1661
Ganoderic acid C2 has anti-inflammatory,and anti-tumor-promoting activities. Ganoderic acid C2 can inhibit histamine release, it also has inhibitory effects on t...
Alginic acid
T20597
Alginic acid (Snow acid algin G) is a natural polysaccharide extracted from brown seaweeds with anti-anaphylactic and anti-inflammatory activities. Alginic acid ...
Chlorphenesin
T4507
Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.
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