T41247 |
Thioperamide maleate
|
148440-81-7
|
98%
|
|
Thioperamide maleate is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31 nM).
|
T1278 |
Astemizole
|
68844-77-9
|
98%
|
|
Astemizole is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors,...
|
T0246 |
Betahistine dihydrochloride
|
5579-84-0
|
98%
|
|
Betahistine hydrochloride is a histamine analog and H1 receptor agonist that serves as a vasodilator.
|
T16759 |
Ritanserin
|
87051-43-2
|
98%
|
|
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adren...
|
T0330 |
Diphenhydramine hydrochloride
|
147-24-0
|
98%
|
|
Diphenhydramine HCl (Benadryl) is a histamine H1 antagonist used as an antitussive and antiemetic. It is also used for pruritus and dermatoses, for hypersensitiv...
|
T1425 |
Pemirolast potassium
|
100299-08-9
|
98%
|
|
Pemirolast Potassium is the potassium salt form of pemirolast, a pyrimidinone derivative with antiallergic property. Pemirolast potassium exerts its action by bl...
|
T0381 |
Amodiaquine dihydrochloride dihydrate
|
6398-98-7
|
98%
|
|
Amodiaquine Hydrochloride is the hydrochloride salt of amodiaquine, an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory properti...
|
T1469 |
Levocetirizine
|
130018-77-8
|
98%
|
|
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
|
T1540 |
Doxepin hydrochloride
|
1229-29-4
|
98%
|
|
Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mech...
|
T1822L |
Clemizole hydrochloride
|
1163-36-6
|
98%
|
|
Clemizole hydrochloride is an antagonist for H1 histamine receptor. According to the research, Clemizole hydrochloride can inhibit hepatitis C virus (HCV) replic...
|
T6488 |
Epinastine hydrochloride
|
108929-04-0
|
98%
|
|
Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
|
T0217L |
(+)-Dropropizine
|
99291-24-4
|
98%
|
|
Levodropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex and by interfering...
|
T0059 |
Diphenylpyraline hydrochloride
|
132-18-3
|
98%
|
|
Diphenylpyraline Hcl is used in the treatment of Parkinsonism.It is a first-generation antihistamine with anticholinergic effects, functions as a dopamine reupta...
|
T0383 |
Fenspiride hydrochloride
|
5053-08-7
|
98%
|
|
Fenspiride, an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use in Russia for the therapy of c...
|
T2232 |
JNJ-7777120
|
459168-41-3
|
98%
|
|
JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM, exhibits >1000-fold selectivity over the other hi...
|
T2335 |
Ebastine
|
90729-43-4
|
98%
|
|
Ebastine (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine. It does not penetrate the blood-brain barrier and thus allows an effe...
|
T2848 |
Osthole
|
484-12-8
|
98%
|
|
Osthole, a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
|
T0217 |
Levodropropizine
|
99291-25-5
|
98%
|
|
Levodropropizine is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
|
T0081 |
Lafutidine
|
118288-08-7
|
98%
|
|
Lafutidine is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.
|
T0211L |
Azelastine hydrochloride
|
79307-93-0
|
98%
|
|
Azelastine Hydrochloride is a phthalazinone derivative with antihistaminergic activity.
|