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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T0031 Ziprasidone hydrochloride monohydrate 138982-67-9 98%
Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
T8822 JNJ-5207852 dihydrochloride 1782228-76-5 98%
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T4499 Mequitazine 29216-28-2 98%
Mequitazine is an effective, nonsedative and long-acting histamine H1 antagonist.
TN1154 Nepetin 520-11-6 98%
6-Methoxyluteolin has antioxidant activity, it is a potent inhibitor of histamine release and calcium influx via down-regulation of the FcεRI α chain.
T1619 Trazodone hydrochloride 25332-39-2 98%
Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depress...
T4099 S 38093 862896-30-8 98%
S-38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
T2533 Alcaftadine 147084-10-4 98%
Alcaftadine is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
T17072 Thiethylperazine dimaleate 1179-69-7 98%
Thiethylperazine dimaleate is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 and possesses antimicrobial, ...
T19443L N-Acetylhistamine acetate 98%
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
T16476 PF-03654746 935840-31-6 98%
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
Ziprasidone hydrochloride monohydrate
T0031
Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
JNJ-5207852 dihydrochloride
T8822
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
Mequitazine
T4499
Mequitazine is an effective, nonsedative and long-acting histamine H1 antagonist.
Nepetin
TN1154
6-Methoxyluteolin has antioxidant activity, it is a potent inhibitor of histamine release and calcium influx via down-regulation of the FcεRI α chain.
Trazodone hydrochloride
T1619
Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depress...
S 38093
T4099
S-38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Alcaftadine
T2533
Alcaftadine is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
Thiethylperazine dimaleate
T17072
Thiethylperazine dimaleate is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 and possesses antimicrobial, ...
N-Acetylhistamine acetate
T19443L
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
PF-03654746
T16476
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
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