T12228 |
Niperotidine
|
84845-75-0
|
98%
|
|
Niperotidine is an antagonist of histamine H2-receptor.
|
T2S0118 |
Daurinoline
|
2831-75-6
|
98%
|
|
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
|
T12703 |
ReN-1869 hydrochloride
|
170149-76-5
|
98%
|
|
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
|
T12416 |
PF-03654746 Tosylate
|
1039399-17-1
|
98%
|
|
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
|
T17118 |
Toreforant
|
952494-46-1
|
98%
|
|
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
|
T15722 |
Lavoltidine
|
76956-02-0
|
98%
|
|
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
|
T11088 |
Doxepin D3 Hydrochloride
|
347840-07-7
|
98%
|
|
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
|
TN2155 |
Rhodiocyanoside A
|
168433-86-1
|
98%
|
|
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
|
T12630 |
(R)-(-)-α-Methylhistamine dihydrobromide
|
868698-49-1
|
98%
|
|
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
|
TN3483 |
Bakkenolide D
|
18456-03-6
|
98%
|
|
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
|
T15590 |
Iodophenpropit dihydrobromide
|
145196-87-8
|
98%
|
|
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
|
T11729 |
JTE-952
|
1255303-54-8
|
98%
|
|
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
|
TN1901 |
(-)-Maackiain
|
2035-15-6
|
98%
|
|
(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
|
T10770 |
Cetirizine D8
|
774596-22-4
|
98%
|
|
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
|
TN3699 |
Corchoionoside C
|
185414-25-9
|
98%
|
|
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
|
T36949 |
Niaprazine
|
27367-90-4
|
98%
|
|
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
|
T21472 |
Dimethindene maleate
|
3614-69-5
|
98%
|
|
Dimethindene maleate is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
|
T0185 |
Escitalopram
|
128196-01-0
|
98%
|
|
Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
|
T15195 |
Ebrotidine
|
100981-43-9
|
98%
|
|
Ebrotidine is a competitive H2-receptor antagonist (Ki: 127.5 nM). It has a potent antisecretory activity and evidenced gastroprotection.
|
T9717 |
Chlorcyclizine
|
82-93-9
|
98%
|
|
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
|