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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T10575 BMY-25271 78441-82-4 98%
BMY-25271
BMY-25271 is an antagonist of histamine H2 receptor.
T11532 H4R antagonist 1 1429375-54-1 98%
H4R antagonist 1
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
T19234 Cetirizine D8 dihydrochloride 2070015-04-0 98%
Cetirizine D8 dihydrochloride
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
TN5279 Zeorin 22570-53-2 98%
Zeorin
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
T12756 ROS 234 dioxalate 1781941-93-2 98%
ROS 234 dioxalate
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
T13040 SUN 1334H 607736-84-5 98%
SUN 1334H
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
T11531 H3R-IN-1 Hydrochloride 2319790-07-1 98%
H3R-IN-1 Hydrochloride
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
T21360 Asenapine 65576-45-6 98%
Asenapine
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, dopamine receptor, and histamine receptor antagonist with antipsychotic effects that is used to tre...
TN1913 Marmin 14957-38-1 98%
Marmin
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
T10769 Cetirizine D4 1219803-84-5 98%
Cetirizine D4
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN3062 4'-O-Methylnyasol 79004-25-4 98%
4'-O-Methylnyasol
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
T19604 WZ4141 1222776-76-2 98%
WZ4141
WZ4141 is an intermediate in compound synthesis.
T12054 MK-0249 862309-06-6 98%
MK-0249
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
T11324 FRG8701 108498-50-6 98%
FRG8701
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
TN2895 3,5-Dicaffeoyl-epi-quinic acid 879305-14-3 98%
3,5-Dicaffeoyl-epi-quinic acid
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
T10911 H3 receptor antagonist 1 935840-13-4 98%
H3 receptor antagonist 1
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
T15565 Imetit dihydrobromide 32385-58-3 98%
Imetit dihydrobromide
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
T4099 S 38093 862896-30-8 99.98%
S 38093
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
T1619 Trazodone hydrochloride 25332-39-2 99.98%
Trazodone hydrochloride
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
T4499 Mequitazine 29216-28-2 99.95%
Mequitazine
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
BMY-25271
T10575
BMY-25271 is an antagonist of histamine H2 receptor.
H4R antagonist 1
T11532
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
Cetirizine D8 dihydrochloride
T19234
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
Zeorin
TN5279
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
ROS 234 dioxalate
T12756
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
SUN 1334H
T13040
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
H3R-IN-1 Hydrochloride
T11531
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
Asenapine
T21360
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, dopamine receptor, and histamine receptor antagonist with antipsychotic effects that is used to tre...
Marmin
TN1913
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
Cetirizine D4
T10769
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
4'-O-Methylnyasol
TN3062
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
WZ4141
T19604
WZ4141 is an intermediate in compound synthesis.
MK-0249
T12054
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
FRG8701
T11324
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
3,5-Dicaffeoyl-epi-quinic acid
TN2895
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
H3 receptor antagonist 1
T10911
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
Imetit dihydrobromide
T15565
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
S 38093
T4099
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Trazodone hydrochloride
T1619
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
Mequitazine
T4499
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
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TargetMol