T10575 |
BMY-25271
|
78441-82-4
|
98%
|
|
BMY-25271 is an antagonist of histamine H2 receptor.
|
T11532 |
H4R antagonist 1
|
1429375-54-1
|
98%
|
|
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
|
T19234 |
Cetirizine D8 dihydrochloride
|
2070015-04-0
|
98%
|
|
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
|
TN5279 |
Zeorin
|
22570-53-2
|
98%
|
|
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
|
T12756 |
ROS 234 dioxalate
|
1781941-93-2
|
98%
|
|
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
|
T13040 |
SUN 1334H
|
607736-84-5
|
98%
|
|
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
|
T11531 |
H3R-IN-1 Hydrochloride
|
2319790-07-1
|
98%
|
|
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
|
T21360 |
Asenapine
|
65576-45-6
|
98%
|
|
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, dopamine receptor, and histamine receptor antagonist with antipsychotic effects that is used to tre...
|
TN1913 |
Marmin
|
14957-38-1
|
98%
|
|
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
|
T10769 |
Cetirizine D4
|
1219803-84-5
|
98%
|
|
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
|
TN3062 |
4'-O-Methylnyasol
|
79004-25-4
|
98%
|
|
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
|
T19604 |
WZ4141
|
1222776-76-2
|
98%
|
|
WZ4141 is an intermediate in compound synthesis.
|
T12054 |
MK-0249
|
862309-06-6
|
98%
|
|
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
|
T11324 |
FRG8701
|
108498-50-6
|
98%
|
|
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
|
TN2895 |
3,5-Dicaffeoyl-epi-quinic acid
|
879305-14-3
|
98%
|
|
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
|
T10911 |
H3 receptor antagonist 1
|
935840-13-4
|
98%
|
|
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
|
T15565 |
Imetit dihydrobromide
|
32385-58-3
|
98%
|
|
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
|
T4099 |
S 38093
|
862896-30-8
|
99.98%
|
|
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
|
T1619 |
Trazodone hydrochloride
|
25332-39-2
|
99.98%
|
|
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
|
T4499 |
Mequitazine
|
29216-28-2
|
99.95%
|
|
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
|