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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T12228 Niperotidine 84845-75-0 98%
Niperotidine is an antagonist of histamine H2-receptor.
T2S0118 Daurinoline 2831-75-6 98%
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12703 ReN-1869 hydrochloride 170149-76-5 98%
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T12416 PF-03654746 Tosylate 1039399-17-1 98%
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T17118 Toreforant 952494-46-1 98%
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T15722 Lavoltidine 76956-02-0 98%
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T11088 Doxepin D3 Hydrochloride 347840-07-7 98%
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
TN2155 Rhodiocyanoside A 168433-86-1 98%
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T12630 (R)-(-)-α-Methylhistamine dihydrobromide 868698-49-1 98%
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN3483 Bakkenolide D 18456-03-6 98%
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T15590 Iodophenpropit dihydrobromide 145196-87-8 98%
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
T11729 JTE-952 1255303-54-8 98%
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
TN1901 (-​)​-Maackiain 2035-15-6 98%
(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
T10770 Cetirizine D8 774596-22-4 98%
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN3699 Corchoionoside C 185414-25-9 98%
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T36949 Niaprazine 27367-90-4 98%
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
T21472 Dimethindene maleate 3614-69-5 98%
Dimethindene maleate is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
T0185 Escitalopram 128196-01-0 98%
Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
T15195 Ebrotidine 100981-43-9 98%
Ebrotidine is a competitive H2-receptor antagonist (Ki: 127.5 nM). It has a potent antisecretory activity and evidenced gastroprotection.
T9717 Chlorcyclizine 82-93-9 98%
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
Niperotidine
T12228
Niperotidine is an antagonist of histamine H2-receptor.
Daurinoline
T2S0118
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
ReN-1869 hydrochloride
T12703
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
PF-03654746 Tosylate
T12416
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
Toreforant
T17118
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
Lavoltidine
T15722
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
Doxepin D3 Hydrochloride
T11088
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
Rhodiocyanoside A
TN2155
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
(R)-(-)-α-Methylhistamine dihydrobromide
T12630
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
Bakkenolide D
TN3483
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
Iodophenpropit dihydrobromide
T15590
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
JTE-952
T11729
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
(-​)​-Maackiain
TN1901
(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
Cetirizine D8
T10770
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
Corchoionoside C
TN3699
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
Niaprazine
T36949
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
Dimethindene maleate
T21472
Dimethindene maleate is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
Escitalopram
T0185
Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
Ebrotidine
T15195
Ebrotidine is a competitive H2-receptor antagonist (Ki: 127.5 nM). It has a potent antisecretory activity and evidenced gastroprotection.
Chlorcyclizine
T9717
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
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