Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T12228	Niperotidine	84845-75-0	98%
T12228	Niperotidine is an antagonist of histamine H2-receptor.
T2S0118	Daurinoline	2831-75-6	98%
T2S0118	Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12703	ReN-1869 hydrochloride	170149-76-5	98%
T12703	ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T12416	PF-03654746 Tosylate	1039399-17-1	98%
T12416	PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T17118	Toreforant	952494-46-1	98%
T17118	Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T15722	Lavoltidine	76956-02-0	98%
T15722	Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T11088	Doxepin D3 Hydrochloride	347840-07-7	98%
T11088	Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
TN2155	Rhodiocyanoside A	168433-86-1	98%
TN2155	Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T12630	(R)-(-)-α-Methylhistamine dihydrobromide	868698-49-1	98%
T12630	(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN3483	Bakkenolide D	18456-03-6	98%
TN3483	Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T15590	Iodophenpropit dihydrobromide	145196-87-8	98%
T15590	Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
T11729	JTE-952	1255303-54-8	98%
T11729	JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
TN1901	(-)-Maackiain	2035-15-6	98%
TN1901	(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
T10770	Cetirizine D8	774596-22-4	98%
T10770	Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN3699	Corchoionoside C	185414-25-9	98%
TN3699	Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T36949	Niaprazine	27367-90-4	98%
T36949	Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
T21472	Dimethindene maleate	3614-69-5	98%
T21472	Dimethindene maleate is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
T0185	Escitalopram	128196-01-0	98%
T0185	Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
T15195	Ebrotidine	100981-43-9	98%
T15195	Ebrotidine is a competitive H2-receptor antagonist (Ki: 127.5 nM). It has a potent antisecretory activity and evidenced gastroprotection.
T9717	Chlorcyclizine	82-93-9	98%
T9717	CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.