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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
TQ0046 Bavisant 929622-08-2 98%
Bavisant is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefulness and cogni...
T0965 Histamine 51-45-6 98%
Histamine is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscl...
T0076 Paliperidone 144598-75-4 98%
Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the pr...
T3979 Emedastine 87233-61-2 98%
Emedastine is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histami...
T19443 N-Acetylhistamine 673-49-4 98%
N-Acetylhistamine is a metabolite of histamine.
T13352 Wy 49051 113418-56-7 98%
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
T4196 Betahistine EP Impurity C 5452-87-9 98%
NSC19005 is structurally related to Betahistine. NSC19005 is a dimer of Betahistine.
T7524 Metiamide 34839-70-8 98%
Metiamide is a histamine H2-receptor antagonist .
T7413 JNJ-5207852 398473-34-2 98%
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T1182 Levocarnitine propionate hydrochloride 119793-66-7 98%
Propionyl-L-carnitine hydrochloride is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudication, and ot...
T20884 Hydroxyzine 68-88-2 98%
Hydroxyzine is an antagonist of histamine H1-receptor.
T6164 Ciproxifan 184025-18-1 98%
Ciproxifan is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
T1045 Trimipramine maleate 521-78-8 98%
Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin an...
T22624L Carcinine ditrifluoroacetate Acetate 98%
Carcinine ditrifluoroacetate is an H3 receptor antagonist.
T11095L DREADD agonist 21 56296-18-5 98%
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T11723L JNJ-39758979 1046447-90-8 98%
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
T31195 Dalcotidine 120958-90-9 98%
Dalcotidine is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to gu...
T0785 Dexchlorpheniramine Maleate 2438-32-6 98%
Dexchlorpheniramine (trade name Polaramine) is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria....
T22842 HTMT dimaleate 195867-54-0 98%
H1 and H2 receptor agonist
TQ0066 GSK189254A 720690-73-3 98%
GSK189254A is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
Bavisant
TQ0046
Bavisant is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefulness and cogni...
Histamine
T0965
Histamine is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscl...
Paliperidone
T0076
Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the pr...
Emedastine
T3979
Emedastine is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histami...
N-Acetylhistamine
T19443
N-Acetylhistamine is a metabolite of histamine.
Wy 49051
T13352
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
Betahistine EP Impurity C
T4196
NSC19005 is structurally related to Betahistine. NSC19005 is a dimer of Betahistine.
Metiamide
T7524
Metiamide is a histamine H2-receptor antagonist .
JNJ-5207852
T7413
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
Levocarnitine propionate hydrochloride
T1182
Propionyl-L-carnitine hydrochloride is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudication, and ot...
Hydroxyzine
T20884
Hydroxyzine is an antagonist of histamine H1-receptor.
Ciproxifan
T6164
Ciproxifan is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
Trimipramine maleate
T1045
Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin an...
Carcinine ditrifluoroacetate Acetate
T22624L
Carcinine ditrifluoroacetate is an H3 receptor antagonist.
DREADD agonist 21
T11095L
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
JNJ-39758979
T11723L
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
Dalcotidine
T31195
Dalcotidine is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to gu...
Dexchlorpheniramine Maleate
T0785
Dexchlorpheniramine (trade name Polaramine) is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria....
HTMT dimaleate
T22842
H1 and H2 receptor agonist
GSK189254A
TQ0066
GSK189254A is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
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