TQ0046 |
Bavisant
|
929622-08-2
|
98%
|
|
Bavisant is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefulness and cogni...
|
T0965 |
Histamine
|
51-45-6
|
98%
|
|
Histamine is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscl...
|
T0076 |
Paliperidone
|
144598-75-4
|
98%
|
|
Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the pr...
|
T3979 |
Emedastine
|
87233-61-2
|
98%
|
|
Emedastine is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histami...
|
T19443 |
N-Acetylhistamine
|
673-49-4
|
98%
|
|
N-Acetylhistamine is a metabolite of histamine.
|
T13352 |
Wy 49051
|
113418-56-7
|
98%
|
|
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
|
T4196 |
Betahistine EP Impurity C
|
5452-87-9
|
98%
|
|
NSC19005 is structurally related to Betahistine. NSC19005 is a dimer of Betahistine.
|
T7524 |
Metiamide
|
34839-70-8
|
98%
|
|
Metiamide is a histamine H2-receptor antagonist .
|
T7413 |
JNJ-5207852
|
398473-34-2
|
98%
|
|
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
|
T1182 |
Levocarnitine propionate hydrochloride
|
119793-66-7
|
98%
|
|
Propionyl-L-carnitine hydrochloride is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudication, and ot...
|
T20884 |
Hydroxyzine
|
68-88-2
|
98%
|
|
Hydroxyzine is an antagonist of histamine H1-receptor.
|
T6164 |
Ciproxifan
|
184025-18-1
|
98%
|
|
Ciproxifan is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
|
T1045 |
Trimipramine maleate
|
521-78-8
|
98%
|
|
Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin an...
|
T22624L |
Carcinine ditrifluoroacetate Acetate
|
|
98%
|
|
Carcinine ditrifluoroacetate is an H3 receptor antagonist.
|
T11095L |
DREADD agonist 21
|
56296-18-5
|
98%
|
|
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
|
T11723L |
JNJ-39758979
|
1046447-90-8
|
98%
|
|
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
|
T31195 |
Dalcotidine
|
120958-90-9
|
98%
|
|
Dalcotidine is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to gu...
|
T0785 |
Dexchlorpheniramine Maleate
|
2438-32-6
|
98%
|
|
Dexchlorpheniramine (trade name Polaramine) is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria....
|
T22842 |
HTMT dimaleate
|
195867-54-0
|
98%
|
|
H1 and H2 receptor agonist
|
TQ0066 |
GSK189254A
|
720690-73-3
|
98%
|
|
GSK189254A is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
|