Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T2848	Osthole	484-12-8	99.87%
T2848	Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
T1575	Nizatidine	76963-41-2	99.87%
T1575	Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
T24421	LY-2624803	879409-35-5	99.87%
T24421	LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.
T20712	Conessine	546-06-5	99.86%
T20712	Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
T6405	Bepotastine Besilate	190786-44-8	99.86%
T6405	Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
T2533	Alcaftadine	147084-10-4	99.86%
T2533	Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
T8514	LML134	1542135-76-1	99.86%
T8514	LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
T4551	Acrivastine	87848-99-5	99.85%
T4551	Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
T21014	Thonzylamine hydrochloride	63-56-9	99.84%
T21014	Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.
T19966	Clemastine	15686-51-8	99.83%
T19966	Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
T22879	JNJ 10191584 maleate	869497-75-6	99.82%
T22879	JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM). JNJ 10191584 maleate inhibits chemotaxis of eosi...
T4566	Lodoxamide	53882-12-5	99.81%
T4566	Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.
T2222	Carbinoxamine Maleate Salt	3505-38-2	99.81%
T2222	Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
T0147	Clemastine fumarate	14976-57-9	99.8%
T0147	Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T2200	Hydroxyzine dihydrochloride	2192-20-3	99.79%
T2200	Hydroxyzine dihydrochloride (Hydroxyzine 2HCl) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and his...
T32191	Irdabisant	1005402-19-6	99.77%
T32191	Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R...
T0118	Mizolastine	108612-45-9	99.77%
T0118	Mizolastine (SL 850324) (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergi...
T0092	Antazoline hydrochloride	2508-72-7	99.76%
T0092	Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous ...
T7893	Bepotastine	125602-71-3	99.75%
T7893	Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.
T22354	Levocetirizine Dihydrochloride	130018-87-0	99.75%
T22354	Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specificall...