Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T0468	Lidocaine	137-58-6	99.74%
T0468	Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation o...
T7085	Mebhydrolin	524-81-2	99.73%
T7085	Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
T26690	AVN-101	1061354-48-0	99.73%
T26690	AVN-101 is a potent 5-HT7 receptor antagonist.
T7176	Pitolisant hydrochloride	903576-44-3	99.72%
T7176	Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
T0942	Quinacrine dihydrochloride	69-05-6	99.72%
T0942	Quinacrine dihydrochloride (Mepacrine dihydrochloride) is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and...
T0162	Quetiapine	111974-69-7	99.71%
T0162	Quetiapine (ICI204636) is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism ...
T2232	JNJ-7777120	459168-41-3	99.71%
T2232	JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM, exhibits >1000-fold selectivity over the other hi...
T1327	Nortriptyline hydrochloride	894-71-3	99.71%
T1327	Nortriptyline hydrochloride (ELF-101 hydrochloride) is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major...
T0074	Chlorprothixene	113-59-7	99.69%
T0074	Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
T68122	Oxmetidine	72830-39-8	99.67%
T68122	Oxmetidine (SKF 92994) is a novel H2 receptor antagonist that is cytotoxic. Oxmetidine inhibits transmembrane calcium flux in cardiac and vascular tissues and is...
T19680	Zotepine	26615-21-4	99.67%
T19680	Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM, 3...
T1553	Chlorpheniramine maleate	113-92-8	99.67%
T1553	Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.
T25875	Noberastine	110588-56-2	99.67%
T25875	Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.
T70489	Enerisant HCl	1152749-07-9	99.66%
T70489	Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins....
T26253	Tecastemizole	75970-99-9	99.66%
T26253	Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
T22240	Amitriptyline	50-48-6	99.64%
T22240	Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties. Amitriptyline is widely used to treat depression and neurop...
T6242	Rupatadine Fumarate	182349-12-8	99.64%
T6242	Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.
T0783	Mianserin hydrochloride	21535-47-7	99.63%
T0783	Mianserin hydrochloride (Org GB 94) is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of...
T1090	Perphenazine	58-39-9	99.63%
T1090	Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0157	Roxatidine Acetate hydrochloride	93793-83-0	99.61%
T0157	Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation....