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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T0211 Azelastine 58581-89-8 99.35%
Azelastine is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
T0137 Mirtazapine 85650-52-8 99.3%
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T68146 Sufotidine 80343-63-1 99.28%
Sufotidine is a highly selective competitive H2 receptor antagonist.
T9084 Cetirizine Impurity B dihydrochloride 1000690-91-4 99.24%
Cetirizine Impurity B dihydrochloride is an impurity of Cetirizine dihydrochloride. Cetirizine is a second-generation antihistamine. Cetirizine is a specific, or...
T22501 2-Pyridylethylamine dihydrochloride 3343-39-3 99.17%
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
T4087 S 38093 HCl 1222097-72-4 99.16%
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
T68056 Donetidine 99248-32-5 99.12%
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
T0445 Promethazine 60-87-7 99.11%
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
T3610 Ranitidine 66357-35-5 99.1%
Ranitidine is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers.
T8548 Metoprine 7761-45-7 99.09%
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
T9770 Samelisant 1394808-82-2 99.09%
Samelisant is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects and can be u...
T1110 Meclizine dihydrochloride 1104-22-9 99.08%
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T10680 Carebastine 90729-42-3 99.06%
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
T3723 Dioxopromethazine hydrochloride 15374-15-9 99%
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
T27244 Efletirizine 150756-35-7 98.98%
Efletirizine is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment of allergic d...
T10000 (±)-Tazifylline 79712-55-3 98.97%
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptor...
T19839 Oxatomide 60607-34-3 98.93%
Oxatomide is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomide can be use...
T1822 Clemizole 442-52-4 98.81%
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
T22842 HTMT dimaleate 195867-54-0 98.51%
H1 and H2 receptor agonist
T27462 GSK-239512 720691-69-0 98.50%
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
Azelastine
T0211
Azelastine is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Sufotidine
T68146
Sufotidine is a highly selective competitive H2 receptor antagonist.
Cetirizine Impurity B dihydrochloride
T9084
Cetirizine Impurity B dihydrochloride is an impurity of Cetirizine dihydrochloride. Cetirizine is a second-generation antihistamine. Cetirizine is a specific, or...
2-Pyridylethylamine dihydrochloride
T22501
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
S 38093 HCl
T4087
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
Donetidine
T68056
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Promethazine
T0445
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
Ranitidine
T3610
Ranitidine is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers.
Metoprine
T8548
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
Samelisant
T9770
Samelisant is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects and can be u...
Meclizine dihydrochloride
T1110
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
Carebastine
T10680
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Dioxopromethazine hydrochloride
T3723
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
Efletirizine
T27244
Efletirizine is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment of allergic d...
(±)-Tazifylline
T10000
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptor...
Oxatomide
T19839
Oxatomide is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomide can be use...
Clemizole
T1822
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
HTMT dimaleate
T22842
H1 and H2 receptor agonist
GSK-239512
T27462
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
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